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1-[(2,5-difluorophenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
1-[(4aR,8aS)-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-6-yl]-2-(3-fluorophenyl)ethan-1-one
N-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2-chlorophenyl)-3-{1-[1-(3-methoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3,5,7-trimethyl-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-N-propyl-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
5-hydroxy-N-{[1-(oxan-4-yl)pyrrolidin-3-yl]methyl}pyrazine-2-carboxamide
1-(4-chlorophenyl)-2-(2,3,4-trimethoxyphenyl)-1H-imidazole
4-[(dimethylamino)methyl]-1-{[3-(trifluoromethoxy)phenyl]methyl}azepan-4-ol
5-({[3-(2-methoxyphenyl)phenyl]formamido}methyl)-N-methylfuran-2-carboxamide
(1R,5S,6S)-6-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-cyclobutylacetamide
4-methyl-2-[4-(2-methylpyridin-4-yl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
2-{methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amino}-2-(thiophen-3-yl)acetic acid
7-(3,4-dimethoxyphenyl)-4-(furan-3-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(1H-indol-3-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]butan-1-one
1-(2-methoxyethyl)-4-[({4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}amino)methyl]pyrrolidin-2-one
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
6-[2,2-bis(prop-2-en-1-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-ethoxy-5-(2-pentylpyrimidin-4-yl)benzoic acid
4-(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}azetidin-3-yl)morpholine
6-methoxy-N-[2-(methylsulfamoyl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[2-(2,2-diphenylethyl)morpholin-4-yl]but-3-en-1-one
4-[1-(6-methoxypyridin-3-yl)-1H-imidazol-2-yl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-(1H-imidazol-1-yl)-1-(thiophene-2-sulfonyl)piperidine-4-carboxylic acid
N-(2,5-dimethyl-3-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}-1H-pyrrol-1-yl)acetamide
8-[(2-chlorophenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-benzoyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
3-chloro-6-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]pyridine-2-carboxylic acid
2,3-dimethyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1H-indole-5-carboxamide
2-benzyl-6-methyl-5-[5-(3-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
(2S)-3-cyclohexyl-2-({1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}amino)propan-1-ol
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-2-propyl-1,3-thiazole-4-carboxamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-4-[(4-fluorophenyl)methyl]piperazine-1-carboxamide
3-({1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidin-3-yl}methyl)benzamide
2-[ethyl({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
2-(dimethylamino)-2-(4-methylphenyl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-(3-chlorophenyl)-2-hydroxy-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
3-{5-[2-(1H-1,2,4-triazol-3-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-amino-4,6-bis(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]morpholine
5-{4-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
2-[(3-fluoropyridin-4-yl)methyl]-2,8-diazaspiro[4.5]decane
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H-pyrazole-4-carboxamide
(4S)-1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}amine
3-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea