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N-(3-fluoro-2-methylphenyl)-2-{4-[2-(thiophen-2-yl)acetyl]morpholin-3-yl}acetamide
2-({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}amino)propan-1-ol
2-(2,4-dichlorophenoxy)-1-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
7-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-(1-carbamoylcyclopentyl)-7-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
3-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methoxyethyl)pyrrolidin-3-yl]-4-methyl-1H-pyrazole-5-carboxamide
2-[2-(dimethylamino)ethyl]-9-{[6-(dimethylamino)pyridin-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-({[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]carbamoyl}methyl)-1H-indole-3-carboxamide
2-(cyclopent-2-en-1-yl)-1-[2-methyl-4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{3-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}acetamide
N-(1-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
2-[(dimethylamino)methyl]-4-[1-(2-methoxyphenyl)-1H-imidazol-2-yl]phenol
4-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]thiomorpholine
3-{2-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(1S,5R)-3-(3-methoxypropyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(1H-pyrazol-1-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine-4-carboxylic acid
6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
N-[(1-{[2-(benzyloxy)phenyl]methyl}piperidin-3-yl)methyl]acetamide
N-[(3-methoxyphenyl)methyl]-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{2-[(3,4,7-trimethyl-1H-indol-2-yl)formamido]acetamido}propanoic acid
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-2-ethylpyrimidine
N-[(2-fluorophenyl)methyl]-3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}propanamide
1-(5-methoxy-2-{[4-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
(1S,5R)-3-(6-methyl-2-propylpyrimidin-4-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-(4-chlorophenyl)-4-(6-methoxypyrimidin-4-yl)morpholine
N,N-dimethyl-6-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]pyrimidin-4-amine
2-(1H-imidazol-2-yl)-1-(propan-2-yl)-1H-1,3-benzodiazole
2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-5-chlorobenzoic acid
2-(phenoxymethyl)-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
(1S,2S)-2-(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-1-yl)cyclohexan-1-ol
4-methyl-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-3,4-dihydro-2H-1,4-benzoxazine
2-(3,4-dichlorophenyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholine
(3S,4R)-1-[1-(dimethylcarbamoyl)piperidine-4-carbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
7-[(2,3-difluorophenyl)methyl]-2-(3-methylbutyl)-2,7-diazaspiro[4.5]decan-6-one
1-(1-{[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-[(3-chlorophenyl)methyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-[(3,3-diethylpyrrolidin-1-yl)methyl]-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N-(pyridin-4-ylmethyl)-1-(pyrimidin-2-yl)piperidin-3-amine
1-{2-[1-(2-hydroxybutyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
2-(4-fluorobenzoyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-fluoro-N-(furan-2-ylmethyl)benzamide
4-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)propane-2-sulfonamide