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3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-[4-({[1-(dimethyl-1,3-thiazol-2-yl)propyl]carbamoyl}amino)phenyl]-N-methylacetamide
7-methyl-2-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
3-(1H-1,3-benzodiazol-2-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
4-(5-methylpyridin-2-yl)-1-phenylmethanesulfonylpiperidin-4-ol
ethyl 4-(3-phenylpropyl)-1-(thiophene-3-carbonyl)piperidine-4-carboxylate
8-[2-(1-ethylpiperidin-4-yl)acetyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(methylsulfanyl)phenyl]-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
ethyl 1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
1-ethyl-N-(2-hydroxyethyl)-5-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-methylthiophene-2-carboxamide
3-cyclohexyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(4-methyl-6-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidin-2-yl)phenol
(3aR,5R,6S,7aS)-2-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-octahydro-1H-isoindole-5,6-diol
5-({[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}methyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-chloro-3-fluoro-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrimidin-2-amine
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[1-(1H-imidazol-1-yl)propan-2-yl]amine
4-methyl-2-({3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,3-thiazole
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrrole-2-carboxamide
4-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]methyl}benzonitrile
2-(dimethylamino)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(3-methylphenyl)acetamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methylphenyl)methyl]amine
2-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine-3-carbonyl}pyridine
2-{[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amino}-N-(pyrazin-2-yl)acetamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
methyl 4-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butanoate
1-(cyclobutylmethyl)-3-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-3-hydroxypiperidin-2-one
N-(1H-imidazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
{3-ethyl-1-[(5-methylpyrazin-2-yl)methyl]piperidin-3-yl}methanol
8-methoxy-N-[2-(methylsulfamoyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
ethyl 1-(pyridin-2-ylmethyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
3-({5-[(E)-2-(4-fluorophenyl)ethenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]propan-1-one
(2S,4S)-4-amino-1-(4-cyanobenzenesulfonyl)-N-methylpyrrolidine-2-carboxamide
4-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
methyl 4-(4-{[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]carbamoyl}piperidin-1-yl)-4-oxobutanoate
(3R,5S)-N-(4-fluorophenyl)-1-(2-methylpropyl)-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
3-methoxy-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
1-[cyclohexyl(methyl)amino]-3-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
[(3R,4R)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
N-[3-(3-ethylphenoxy)propyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-{2-[(prop-2-en-1-yl)amino]benzoyl}azetidin-3-ol
4-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)-1H-pyrazole-3-carboxylic acid
1-[(4-fluorophenyl)methyl]-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
3-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,3-oxazolidin-2-one