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1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-phenylpyrimidin-2-amine
5-(2-methoxyphenoxymethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
(2R,6R)-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
3-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,2-dihydroquinolin-2-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
1-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
2-({[3-hydroxy-2-oxo-1-(3-phenylpropyl)piperidin-3-yl]methyl}amino)-N,N-dimethylacetamide
4-(naphthalen-2-ylmethyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[2-(2-chloro-6-fluorophenyl)acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-hydroxyethyl)-N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
(benzylsulfamoyl)[2-(3,4-dimethoxyphenyl)ethyl]methylamine
1-[2-(3,5-dimethoxyphenyl)-2-hydroxyethyl]-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
N-[(2-methoxyphenyl)methyl]-2-{[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}-N-(prop-2-en-1-yl)acetamide
5-hydroxy-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]pyrazine-2-carboxamide
1-(diethylamino)-3-(2-methoxy-4-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}phenoxy)propan-2-ol
4-{[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(oxolane-3-carbonyl)piperidine
3-[(3R,4S)-3-(2-amino-4-ethyl-1,3-thiazole-5-amido)-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
2-[methyl({4-methyl-5-[1-(pyridine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-benzylpiperidin-4-yl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-methylacetamide
2-[4-(1-benzothiophen-3-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[(3S,4R)-1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(1H-imidazol-4-ylmethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
1-(6-{methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}pyridin-2-yl)ethan-1-ol
6-[4-(1,3-thiazol-2-yl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
4-ethyl-3-{1-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,7aS)-1-(2-{[3-(dimethylamino)propyl](methyl)amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-4-yl)ethan-1-one
6-methyl-3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
3,5-dimethyl-1-(1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidin-3-yl)-1H-pyrazole
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
3-cyclopropyl-5-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazol-3-yl]-1-phenyl-1H-1,2,4-triazole
2-(2-methoxyphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N'-(3-chloro-2-methylphenyl)-N-[1-(hydroxymethyl)cyclopentyl]propanediamide
2-hydroxy-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3,5-bis(propan-2-yl)benzamide
4-[1-(2-phenylethyl)pyrrolidin-3-yl]-1-[1-(trifluoromethyl)cyclopropanecarbonyl]piperidine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[3-(dimethylamino)pyrrolidin-1-yl]pyridine-3-carboxamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(5-oxopyrrolidine-3-carbonyl)-1,4-diazepan-2-one
3-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1,2-dihydropyridin-2-one
(2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)urea
4-{1-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethyl}-2-fluorophenol
(4aS,8aR)-6-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-methanesulfonyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
diethyl[(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5-phenylfuran-2-yl)methyl]amine
methyl (2S,4S)-1-methyl-4-[3-(1,2-oxazinan-2-yl)propanamido]pyrrolidine-2-carboxylate
N-[(2-fluorophenyl)methyl]-5-[(3-hydroxypropyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide