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2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-1-ol
4-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}piperazin-2-one
2-(3-{[(2-methoxyethyl)(1-methylpiperidin-4-yl)carbamoyl]amino}phenyl)acetamide
N-methyl-N-(2-phenylethyl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
(1R,2R,6S,7S)-N-(7-chloro-2-ethyl-3-methyl-1-benzofuran-5-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
5-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-(2-methoxyphenyl)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
2-(2-phenylethyl)-4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}morpholine
N-(2,4-dimethylphenyl)-3-(4-methyl-1,4-diazepan-1-yl)-3-oxopropanamide
4-[3-(4-benzylpiperidine-1-carbonyl)piperidin-1-yl]-2-(2-methoxy-2-methylpropyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-tert-butyl-6-(2,5-dimethoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
4-methoxy-6-[(2S)-2,4,5,5-tetramethylpiperazin-1-yl]pyrimidine
(1R,5S,6R)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methylphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
(4aR,7aS)-1-acetyl-4-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(furan-2-ylmethyl)piperidine-3-carboxamide
2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2,3-dihydro-1H-isoindole
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-4-hydroxypiperidine-4-carboxylic acid
2-(2-methoxyphenoxy)-N-{[1-(pyrazine-2-carbonyl)piperidin-3-yl]methyl}acetamide
5-amino-2-ethyl-1-(3-methoxypropyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-{3-[4-({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)piperidin-1-yl]phenyl}cyclopropanecarboxamide
5-[4-(3-methoxypropyl)piperidine-1-carbonyl]-1-(3-phenylpropyl)piperidin-2-one
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[4-(piperidin-3-yl)benzoyl]piperazine
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
4-[(4-methoxyphenyl)methyl]-3-[(4-methylpiperazin-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
(4aR,7aS)-1-cyclopentanecarbonyl-4-(1-methyl-1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2,4,6-trimethyl-3-{[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]methyl}phenyl)methyl acetate
N-ethyl-5-(3-ethylpiperazine-1-carbonyl)-4-methyl-1,3-thiazol-2-amine
N-[(2-methyl-1H-indol-5-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(3-methyl-1H-pyrazole-5-carbonyl)morpholine
N-ethyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
dimethyl(3-{2-[1-(quinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(2-methoxyphenyl)propanamide
N-[(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
(3S,4R)-N,N-dimethyl-4-propyl-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(3-oxopiperazin-1-yl)acetamide
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-1-(3-methoxypropyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
5-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-N-methylfuran-2-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-methanesulfonylpropan-1-one
N-methyl-6-(4-methyl-1,4-diazepan-1-yl)-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
2-methyl-5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
2-{[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-5,8-dimethylquinolin-4-ol