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N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
5-(8-fluoroquinoline-2-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
5-phenyl-2-(pyridin-4-yl)-4-[1-(2,3,6-trifluorobenzoyl)piperidin-3-yl]pyrimidine
2-[4-(4-methylphenyl)piperazin-1-yl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(5-{1-[(2S)-oxolan-2-ylmethyl]-1H-imidazol-2-yl}furan-2-yl)benzonitrile
2-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}benzoic acid
2-(dimethylamino)-N-(2-methoxyethyl)-2-(4-methylphenyl)-N-(pyridin-2-ylmethyl)acetamide
[2-(2,5-difluorophenyl)ethyl](methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
4,6-dimethyl-N-{2-[methyl(phenyl)amino]propyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(4-methylphenyl)methyl]-5-[2-(methylsulfanyl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
3-{2-[(2-ethylpyrimidin-5-yl)formamido]acetamido}propanoic acid
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)thiophene-2-sulfonamide
[(6-methylpyridin-2-yl)methyl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
(1R,5R)-6-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-(1H-pyrazol-1-ylmethyl)-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-3-(pyrazin-2-yl)propanamide
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
N-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]acetamide
1-[(furan-2-ylmethyl)carbamoyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-{2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
(3R,5S)-N-butyl-1-[(3,4-dimethoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-4-(1H-pyrazol-1-yl)butan-1-one
(2S,4S)-4-amino-N-(propan-2-yl)-1-(quinoline-8-sulfonyl)pyrrolidine-2-carboxamide
(1S,5R)-6-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(3R,4S)-1-[2-(3-methoxyphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(2-hydroxypropyl)-9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(prop-2-en-1-yl)propanamide
[(6-chloropyridin-3-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-[N-methyl4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-amido]cyclopentane-1-carboxylic acid
2-(4,6-dimethylpyrimidin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-phenoxy-N-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyrimidin-4-amine
6-[3-(pyridin-2-yl)azetidin-1-yl]-9H-purine
N-(4-fluoro-2-methylphenyl)-3-[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-3-yl]propanamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}azocane
2-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-[1-(3-methoxy-5-methylthiophene-2-carbonyl)piperidin-2-yl]pyridine
3-(5-{[3-(naphthalene-2-carbonyl)piperidin-1-yl]methyl}-1,3,4-oxadiazol-2-yl)pyridine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2,3-dihydro-1-benzofuran-7-carboxamide
7-(4-chlorophenyl)-2-(4-propyl-4H-1,2,4-triazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)piperidine-4-carbonitrile
N-methyl-5-[(methylsulfanyl)methyl]-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]furan-2-carboxamide
2-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
(2-{[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)amino}ethyl)dimethylamine
2-{2-[3-(2-methoxyethyl)-1-methyl-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
1-{3-[4-(benzyloxy)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)pyridine
2-{4-[2-(morpholin-3-yl)acetamido]phenyl}quinoline-4-carboxamide