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3-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
3-cyclopropyl-1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)(quinolin-4-ylmethyl)amine
4-({1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-[2-(2-chlorophenoxy)ethyl]-1-(methoxymethyl)cyclopropane-1-carboxamide
ethyl 2-{methyl[5-({[1-(1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)pyrimidin-2-yl]amino}acetate
N-[2-(2-fluorophenyl)-1-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)ethyl]-N-methylthiophene-2-carboxamide
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
7-(cyclopropylmethyl)-2-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2,7-diazaspiro[4.5]decane
methyl 1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazole-3-carboxylate
1-[(4-methoxyphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
1-(2-aminoethyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclopentanecarbonyl-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[(3-methylphenyl)methyl]-5-(morpholine-4-carbonyl)-1-propyl-1H-1,3-benzodiazol-2-amine
4-(4-chlorophenoxy)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
2-(3-methoxypropyl)-9-[(3-methylquinoxalin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
butyl 2-(pyridin-2-yl)pyrrolidine-1-carboxylate
N-methyl-3-(2-oxopyrrolidin-1-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
2-[3-(oxolan-3-yl)-5-(1-phenyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N'-(2-fluoro-5-methylphenyl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}butanediamide
(4aS,8aR)-1-(3-aminopropyl)-6-(2-aminopyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-phenylethane-1,2-dione
1-(2-amino-9H-purin-6-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[2-oxo-2-(pyridin-3-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
1-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
3-(oxolan-3-yl)-5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]-1H-1,2,4-triazole
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
(2S,4S)-N-ethyl-4-{[(4-methoxy-3-methylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-{[4-(benzyloxy)phenyl]methyl}-3-(1H-pyrazol-5-yl)piperidine
4-{1-[2-(1,1-dioxo-1λ6-thian-4-yl)acetyl]pyrrolidin-3-yl}benzoic acid
1-ethyl-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
8-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
3-[1-(2,2-difluorobutanoyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(methoxymethyl)cyclopentyl]-3-(2-methylphenyl)propanamide
N-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-N-(4-methylphenyl)methanesulfonamide
1-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-(2,3,5-trifluorophenyl)urea
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[2-(pyridin-2-ylmethoxy)phenyl]urea
N-[4-(ethylcarbamoyl)phenyl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
4-(2-methoxyacetyl)-N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-1,4-diazepane-1-carboxamide
[(2,4-difluorophenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
ethyl 2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]acetate
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(2-methylbenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}){[2-(trifluoromethyl)phenyl]methyl}amine
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl]methanol