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8-[(3E)-pent-3-enoyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 3-[(4-fluorophenyl)methyl]-1-(3-methylbutanoyl)piperidine-3-carboxylate
3-(furan-2-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
5-[1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)pyrrolidin-2-yl]-N-methylthiophene-2-carboxamide
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-amino-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
8-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(8-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl)acetic acid
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
2-(3-fluoro-4-hydroxyphenyl)-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}acetamide
2-{1-[(4-ethoxyphenyl)methyl]-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-(2-{4-[1-(4-methylphenyl)piperidin-4-yl]morpholin-2-yl}ethyl)acetamide
3-{5-[4-(1H-pyrazol-3-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-(1'-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
(1R,9aR)-1-[({2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(thiophen-2-ylmethyl)acetamide
N-{4-[(2,6-dimethylphenyl)carbamoyl]phenyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(2-methoxyphenyl)methyl]-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-{3-[3-methyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}acetamide
methyl 3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(1S,2R)-2-aminocyclobutyl]-2-[3-chloro-2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]ethan-1-one
(2S,4S)-4-amino-1-[4-(4-methoxyphenyl)butanoyl]-N-methylpyrrolidine-2-carboxamide
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)phenol
2-(5-oxo-2-phenylcyclopent-1-en-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
3-[({1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
1-{4-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]phenyl}-3-(oxolan-2-ylmethyl)urea
3-(4-benzylpiperazine-1-carbonyl)-1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-1,4-dihydropyridin-4-one
N-{2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylformamido]ethyl}pyridine-3-carboxamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
N-({5-[(5-cyclopentylthiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N-[(3-methoxyphenyl)methyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
3-{3-cyclopropyl-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}pyridine
N,2,7-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
3-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(2-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
2-(dimethylamino)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(3-methylphenyl)acetamide
(1S,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(2,2-diphenylethyl)-3,9-diazabicyclo[3.3.2]decan-10-one
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(propan-2-yloxy)propyl]propanamide
6-ethyl-N2,N2-dimethyl-N4-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidine-2,4-diamine
N-benzyl-2-[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-(thiophen-3-ylmethyl)urea
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-(1H-1,2,4-triazol-3-yl)benzamide
[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
8-(2-amino-6-methylpyrimidin-4-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one