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N-methyl-N-[2-(morpholin-4-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
1-{2-[1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-2-one
2-{1-cyclohexyl-4-[(3-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(2S)-2-amino-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[3-(pyrrolidin-1-yl)propyl]acetamide
1-(4-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-(2-methoxyphenoxy)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)azetidine-1-carboxamide
3-amino-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
1-(4-fluorophenyl)-4-{imidazo[1,2-a]pyridine-6-carbonyl}piperazine
N-ethyl-3-(3-methoxyphenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
(1R,6S)-9-methyl-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propane-1,3-diol
(4aR,8aS)-1-[3-(1H-imidazol-1-yl)propyl]-6-(3-methylthiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]ethan-1-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
ethyl 1-[5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-2-carboxylate
5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-N-phenylpyrimidin-2-amine
(2S)-N2-ethyl-N1-(3-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)pyrrolidine-1,2-dicarboxamide
2-{2-[3-(4-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-8-methyl-2,8-diazaspiro[4.5]decan-3-one
methyl 3-{[7-oxo-4-(thiophene-2-carbonyl)-1,4-diazepan-1-yl]methyl}benzoate
1-(2-methoxyphenyl)-3-{1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
6-methyl-4-oxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4H-pyran-2-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-methyl-4-oxo-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pentanamide
9-(5-acetylpyridin-2-yl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
1-(furan-2-ylmethyl)-4-[5-(hydroxymethyl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N,N-dimethyl-4-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperazine-1-sulfonamide
N,1-dimethyl-5-(4-methylpiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S)-2-(methoxymethyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)pyrrolidine-1-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-(1-methylpyrrolidin-3-yl)pyrimidine-5-carboxamide
(4S)-4-amino-5-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-oxopentanoic acid
1-methyl-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indole
N-{5-[(2S)-2-acetamidopropanamido]-2-methoxyphenyl}benzamide
methyl 5-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-5-oxopentanoate
4-hydroxy-1-(2-phenylquinoline-4-carbonyl)piperidine-4-carboxylic acid
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-3-sulfonamide
N-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
2-[4-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
7-(cyclohexylmethyl)-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(3R)-1-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-ol
N,N-dimethyl-6-(3-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridazin-3-amine
N4-[2-(7-methyl-1H-indol-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-(piperidin-1-yl)-1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidine
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-(naphthalen-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2-methyl-3-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanoic acid