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ethyl(1,3-thiazol-4-ylmethyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2-methylphenyl)methyl]benzamide
5-{[1-(ethoxycarbonyl)cyclobutyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[4-(2-{octahydropyrrolo[1,2-a]piperazin-2-yl}-2-oxoethoxy)phenyl]propan-1-one
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methoxy-1H-indole
5-[2-(2-chloro-6-fluorophenyl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-2-(pyridin-4-yl)quinoline
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-(2-fluorophenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
(5S,9aS,9bS)-2-methyl-5-[4-(2-methylpropyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-3-(pyridin-3-yl)propanamide
8-(2,3-dimethyl-1H-indole-7-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}oxane-2-carboxamide
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]benzonitrile
N-[(2R,3R)-2-methoxy-1'-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(1H-1,2,4-triazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
2-(4-chlorophenyl)-4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]morpholine
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]urea
N-(2,3-dihydroxypropyl)-6-(methoxymethyl)-N-methylpyridine-2-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(3-methoxyphenoxymethyl)piperidine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(oxolan-2-yl)acetamide
3-(benzenesulfonyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
5-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}-N-phenylpyrimidin-2-amine
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-(1H-pyrrole-2-carbonyl)piperazine
1-[(3R,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
N-(4-fluoro-3-methylphenyl)-3-[(6-oxopiperazin-2-yl)formamido]propanamide
4-[4-(3-hydroxyphenyl)-1H-1,2,3-triazol-1-yl]-N,N-dimethylbutanamide
methyl 4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazine-1-carboxylate
3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,N-dimethylpropanamide
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(2-methoxyphenyl)ethan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-8-(2,2-dimethylpropyl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,2-dimethyl-N-(2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethyl)propanamide
6-fluoro-4-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3S,4R)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}cyclobutanamine
2-benzyl-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-cyclohexyl-5-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}pyrimidine
1-[2-(2,5-dimethylphenoxy)ethyl]-5-oxopyrrolidine-3-carboxylic acid
N-cyclopentyl-5-hydroxy-N-(thiophen-3-ylmethyl)pyrazine-2-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-2-{[3-(3-hydroxy-3-methylbutyl)phenyl]formamido}-2-phenylacetamide
3-(2,4-difluorophenyl)-4-{1H-imidazo[4,5-b]pyridin-2-yl}-1H-pyrazole
(3S,4R)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-methylpiperidine-3,4-diol
methyl 2-{7-chloro-3-[(diethylamino)methyl]-2-oxo-1,2-dihydroquinolin-1-yl}acetate
4-[3-(5-methylthiophen-2-yl)-5-(pyrrolidine-1-carbonyl)benzenesulfonyl]morpholine
(4aR,8aR)-4a-hydroxy-7-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide