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2-butyl-8-(1H-indole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-3-(5-methylfuran-2-yl)-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
(2E)-N-{[7-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
(4aS,7aR)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-cyclopropaneamido-4-methyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]benzamide
6-{[1-(3-chlorophenyl)piperidin-4-yl]amino}-2-methylheptan-2-ol
4-[2-(benzyloxy)ethyl]isoquinoline
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-ethyl-7-methyl-N-[2-(3-methylphenoxy)ethyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-{methyl[(3-methylpyridin-2-yl)methyl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(3R,4S)-1-[6-(methoxymethyl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-amine
4-({2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)benzene-1-sulfonamide
2-(3,4-dichlorophenyl)-4-(6-ethylpyrimidin-4-yl)morpholine
5-amino-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1H-pyrazole-3-carboxamide
1-(1-methyl-1H-indole-6-carbonyl)azetidine-2-carboxylic acid
1-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]-3-(1H-pyrazol-5-yl)piperidine
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1,2-oxazole-5-carboxamide
N4-methyl-N4-[4-(morpholin-4-yl)butyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
4-[3-(1-benzofuran-2-yl)phenyl]-4H-1,2,4-triazole
1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
6-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-{2-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-[4-(4-acetylphenyl)piperazin-1-yl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-(4-methylthiophen-2-yl)pyridine-3-carboxamide
3-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-(dimethylamino)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-cyclopropylquinoline-2-carboxamide
1-[2-methoxy-5-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(1-methyl-1H-imidazol-2-yl)[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]methanol
(2S,5R)-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethylpiperazine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-(5-methylfuran-2-yl)benzamide
1-({5-[(4-chloro-3-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
{1-[(3-methylthiophen-2-yl)sulfonyl]-4-(oxan-2-ylmethyl)piperidin-4-yl}methanol
ethyl 3-[5-(1H-pyrazol-1-ylmethyl)furan-2-amido]azepane-1-carboxylate
methyl 3-ethanesulfonamido-5-{[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamido]methyl}benzoate
methyl 2-{[5-(4-fluorophenyl)-4-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
2-{4-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]piperazin-1-yl}pyridine-3-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-imidazole-4-sulfonamide
4-(pyridin-3-ylmethoxy)-N-(trimethyl-1H-pyrazol-4-yl)piperidine-1-carboxamide
methyl (2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]morpholin-3-yl}acetic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-hydroxy-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(4-methoxyphenyl)methyl]-5,6-dimethyl-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
3-[N-(2-phenylethyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]formamido]propanamide
6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-3-carboxamide
2-cyclopropyl-5-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3,4-dihydropyrimidin-4-one
2-[2-(butan-2-yl)phenoxy]-N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
4-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-5-(propan-2-yl)pyrimidine
1-[(2S)-1-acetylpyrrolidine-2-carbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid