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1-(2-methoxyphenyl)-5-methyl-4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperazin-2-one
2-{4-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]phenoxy}acetamide
N,2-diethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
4-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)pyrimidin-2-amine
1'-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]spiro[indene-1,4'-piperidine]
(3R,5S)-N-(2-phenylethyl)-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
N-[1-(propan-2-yl)-1H-pyrazol-4-yl]-4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
N-({1-[(4-fluoro-3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-methoxy-2-methylpropanamide
5-tert-butyl-4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]furan-2-carboxamide
{4-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}methanol
4-(3-hydroxy-3-methylbutyl)-N-[(5-methylpyrazin-2-yl)methyl]benzamide
N'-cyclopentyl-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]butanediamide
4-{1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)-4-phenylbenzamide
(3R,5S)-N-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-(pyridin-4-ylmethyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
1-[2-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
3-(4-ethyl-1H-pyrazol-5-yl)-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperidine
2-(4-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}-6-methylpyrimidin-2-yl)phenol
4-ethyl-1-methyl-3-[(1-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-ethoxynaphthalen-1-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3S,4R)-1-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
8-[5-(hydroxymethyl)furan-2-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methyl-2-phenyl-1-(3-phenyl-1H-pyrazole-4-carbonyl)piperazine
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-{1-[1-(3-phenoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(pyridin-4-ylsulfanyl)acetamide
N-ethyl-3,4-dimethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-5-sulfamoylbenzamide
6-(1-{3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanoyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
5-{4-phenyl-1-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-5-yl}isoquinoline
2-[5-(5-methylpyrazin-2-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-benzyl-9-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-(3,4-dihydroxyphenyl)-6-[4-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[2-(pyridin-3-yloxy)ethyl]acetamide
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-3-carboxamide
5-(3-fluorophenoxymethyl)-3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1H-pyrazole
(2E)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-3-phenylprop-2-enamide
4-(4-methyl-1H-pyrazol-1-yl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidine-4-carboxylic acid
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
(2R,6S)-2,6-dimethyl-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperidine
4-[(benzyloxy)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-2-methyl-1,4-diazepan-5-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
N-[(2R,4R,6S)-2-(propan-2-yl)-6-[1-(propan-2-yl)-1H-pyrazol-4-yl]oxan-4-yl]benzamide
1-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
1-[2-(4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]piperazine
(3R,4R)-3-[(2,3-dihydro-1H-inden-2-yl)amino]-4-hydroxy-N-(2-methylphenyl)pyrrolidine-1-carboxamide
(3S)-4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-ethylmorpholine
3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridin-2-amine