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N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-(3-methoxyphenyl)-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
5-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,3-oxazole-4-carboxamide
2,6,8-trimethyl-4-(3-phenoxyazetidine-1-carbonyl)quinoline
4-[(6-methylpyridin-2-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-{4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-1-yl}pyridine-3-carbonitrile
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-(piperidin-3-ylmethyl)benzamide
4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}thiomorpholine
N-[(2,2-dimethyloxan-4-yl)methyl]-N-(pyridin-2-ylmethyl)cyclopropanamine
1-[1-(5-chloro-2-fluorobenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
3,8-bis[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrrolidine-1-carboxamide
(2R)-2-hydroxy-2-phenyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
(1R,5R)-6-(cyclopropylmethyl)-N-[(2-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
5-{3-[2-(cyclohex-3-en-1-yl)-1H-imidazol-1-yl]propyl}-4-methyl-1,3-thiazole
1-{2-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethan-1-one
3-[5-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[2-(2-ethylphenoxy)ethyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,3-dihydro-1H-isoindole
6-methyl-5-[5-(1-methylpiperidin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[2-(2-chlorophenoxy)ethyl]-1-(thiophene-2-carbonyl)piperidin-4-amine
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
7-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{2-[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1S)-1-phenylethyl]urea
3-phenyl-1-[1-(quinoline-6-carbonyl)piperidin-3-yl]propan-1-one
(3R,5S)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N3-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N3-(2-phenylethyl)-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-({2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}amino)pyridine-3-carbonitrile
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(2-methanesulfonylethyl)piperazine
5-[4-(2,3-dimethylphenyl)piperazin-1-yl]-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
4,4-difluoro-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}piperidine-1-carboxamide
1-methyl-4-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
5-methanesulfonyl-2-methyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
6-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-amine
N-{1-[1-(2,4-difluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-2-methylpropyl}acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)acetamide
4-{2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}morpholine
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
13-(1-benzofuran-2-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-(2,2-dimethyloxan-4-yl)-N-ethyl-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
3-(2,2-dimethylpyrrolidine-1-carbonyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinoxalin-6-ylmethyl)benzamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-3-(1,2-oxazinan-2-yl)propanamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(6-methylpyridin-2-yl)methyl]propanamide
2-(3-{1-[(6-chloropyridin-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-[(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide