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N-[(3R,4R)-3-hydroxy-1-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl]pyridine-2-carboxamide
1-(6-hydroxy-4-methyl-1,4-diazepan-1-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
[1-(1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
1-[(1-{6-[3-(aminomethyl)pyrrolidin-1-yl]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
ethyl 4-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)piperidine-1-carboxylate
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(methylamino)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-[(5-methylfuran-2-yl)methyl]propanamide
3-[4-(dimethylamino)phenyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
4-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]benzamide
2-(2-oxo-1'-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl)acetamide
3-methoxy-6-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridazine
4-(1-benzyl-1H-imidazol-2-yl)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
1-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N,1,7-trimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-indole-2-carboxamide
N-[(1-methyl-1H-imidazol-5-yl)methyl]-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopentanamine
1-{3-[1-(2-hydroxyethyl)-3-(2-methoxyphenoxymethyl)-1H-1,2,4-triazol-5-yl]phenyl}ethan-1-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(morpholin-4-yl)-2-oxoacetamide
methyl[(5-methylfuran-2-yl)methyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(4-hydroxy-2-methylphenyl)pyridine-3-carbonitrile
6-methyl-5-(2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3-chloro-5-fluorophenyl)methyl]-N-(pyridin-4-ylmethyl)cyclopropanamine
4-ethyl-1-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-diethyl-1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
N-(1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}cyclopentyl)-4-methoxyaniline
5-[(dimethylamino)methyl]-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]furan-2-carboxamide
[7-chloro-5-(1-methyl-1H-indazol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-[5-(piperidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aR)-5-[(2,5-difluorophenyl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-4-amino-N-ethyl-1-[1-(2-methoxyphenyl)piperidin-4-yl]pyrrolidine-2-carboxamide
2-(1-methyl-1H-imidazol-2-yl)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine
3-methyl-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
N-(3-carbamoyl-4-fluorophenyl)-4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
4-[(2-chlorophenyl)methyl]-1-(1H-indole-6-carbonyl)-1,4-diazepan-5-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-ethyl-5-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
2-chloro-N-({1-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)benzamide
N-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-5-methyl-1,3,4-oxadiazol-2-amine
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-3-yl)-1,3-thiazole-4-carboxamide
5-amino-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
(2S)-2-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamido]-3-(4-hydroxyphenyl)propanamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
(3R)-1-{1-[3-(furan-2-yl)phenyl]piperidin-4-yl}pyrrolidin-3-ol
2-(1H-indazol-1-yl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
1-{5-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-cyclopentyl-4-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-1,4-diazepan-6-ol
N,2,2-trimethyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)oxan-4-amine