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2-[1-cyclopentyl-4-(quinolin-6-ylmethyl)piperazin-2-yl]ethan-1-ol
2-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}pyridin-3-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(cyclohexylmethyl)amino]-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-methyl-N-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
(2S)-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5-oxopyrrolidine-2-carboxamide
N-[3-(aminomethyl)-5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenyl]pyridine-2-carboxamide
N-(4-chloro-2-methylphenyl)-4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
3-(4-chlorophenyl)-2-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
8-[3-(1H-imidazol-1-yl)propyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-cyclopentyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1H-1,3-benzodiazole-6-carboxylic acid
(2R,3R)-3-(dimethylamino)-1'-(2-ethylpyrimidine-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2,6-dimethoxy-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridine
1-[(4aR,8aS)-1-(quinoxaline-6-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
N-{[1-(6-ethyl-5-fluoropyrimidin-4-yl)piperidin-3-yl]methyl}-2-(4-methoxyphenyl)acetamide
(2S,4R)-4-amino-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-cyclopentyl-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2-phenylacetamide
4-[2-methyl-4-(2-methylphenyl)-5-oxopiperazin-1-yl]-4-oxobutanamide
4-[({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1-methyl-1,2,3,4-tetrahydroquinolin-2-one
1-(4-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}thiophen-2-yl)ethan-1-one
methyl 2-{8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
3-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3H,4H-pyrido[4,3-d]pyrimidin-4-one
5-(2-methoxypyridine-3-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2E)-3-(3-fluorophenyl)-N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}prop-2-enamide
1-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-phenoxypropan-2-ol
3-methyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,2-dihydroquinoxalin-2-one
1-methyl-6-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,6-dihydropyridine-3-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-3-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)propanamide
methyl 4-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]benzoate
2-ethyl-4-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
3-methoxy-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]propanamide
4-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
3-(3-hydroxyquinoxalin-2-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}propanamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-[(2,6-difluorophenyl)methyl]-N-[2-(pyridin-3-yloxy)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-chloro-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2,5-dimethylbenzene-1-sulfonamide
(1S,5R)-6-(2-methylpyrimidine-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-5-({6-oxo-2,7-diazaspiro[4.5]decan-2-yl}sulfonyl)benzoic acid
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-5-methyl-6-phenylpyridine-3-carbonitrile
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1,2,3-thiadiazole-4-carboxamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl](3,3,3-trifluoro-2-methylpropyl)amine
8-(pyridazine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-methoxy-3-(1-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-1,2,3-triazol-4-yl)phenol
N,N-dimethyl-3-[2-({methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)phenyl]propanamide
ethyl 5-benzyl-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]quinoline-4-carboxamide