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(3R,4R)-1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
5-{1-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxylic acid
2-[1-(cyclohexylmethyl)-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
methyl (1R,3S)-3-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]cyclopentane-1-carboxylate
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}piperidin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
(2S,4R)-1-benzyl-N,N-diethyl-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-cyclohexyl-2-(hydroxymethyl)-N-(pyridin-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(4-fluorophenyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,2,3,6-tetrahydropyridine
5-ethyl-4-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-oxazole
4-fluoro-3-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}sulfonyl)benzoic acid
(1S,2R)-N1-[(4-ethylphenyl)methyl]-N1-(2-methoxyethyl)-N2-methylcyclohexane-1,2-dicarboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
4-{5-fluoro-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-4-yl}morpholine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(ethylsulfanyl)propanamide
ethyl 4-[6-oxo-1-(2-phenylethyl)piperidine-3-carbonyl]piperazine-1-carboxylate
1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-[(4aR,7aS)-4-[(2-ethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
[1-(1-methyl-1H-pyrazol-5-yl)propyl]({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)amine
2-{4-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
({5-[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)dimethylamine
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(2-phenoxyethyl)piperidine-4-carboxamide
4-phenoxy-1-(pyridin-4-yl)piperidine-4-carboxylic acid
3-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
2'-amino-4'-(furan-2-yl)-7',8'-dihydro-5'H-spiro[piperidine-4,6'-quinoline]-3'-carbonitrile
(1S,5R)-3-(2-chloro-5-methylbenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-tert-butyl-5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-yl)-3-(furan-2-yl)-1H-1,2,4-triazole
[(3S,5R)-1-(3-chloro-5-methoxybenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
2-{4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperazin-1-yl}-N,N-dimethylacetamide
3-(dimethylsulfamoyl)-N-[3-(1H-imidazol-1-yl)propyl]-5-[(thiophen-3-ylmethyl)amino]benzamide
1-cyclopentyl-N-(1H-indol-6-ylmethyl)-5-oxopyrrolidine-3-carboxamide
1-benzyl-N-ethyl-5-[(2-methoxyethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methoxyphenyl)ethan-1-one
2-butanoyl-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
8-[(6-chloro-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-hydroxy-N-[2-(2-phenoxyethoxy)phenyl]benzamide
(3S,4R)-3-cyclopropyl-N,N-dimethyl-4-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamido]pyrrolidine-1-carboxamide
N-(2-{1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]piperidin-3-yl}ethyl)acetamide
6-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
6-(methoxymethyl)-N-{[1-(methoxymethyl)cyclopentyl]methyl}pyrimidin-4-amine
3-{[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}benzoic acid
5-{imidazo[1,2-a]pyrimidin-6-ylmethyl}-3-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-{2-[2-(1H-pyrazol-1-yl)benzoyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
4-(benzyloxy)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
2-[2-(adamantan-1-ylsulfanyl)acetamido]-N,N-dimethylpropanamide
6-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-({2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-ethyl-N4-[2-(pyridin-3-yloxy)propyl]pyrimidine-2,4-diamine
6-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]pyridine-3-carbonitrile