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N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-4-methylbenzamide
3-(furan-2-ylmethyl)-3-(1-hydroxybutan-2-yl)-1-(4-methanesulfonylphenyl)urea
N2-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-methylpyrimidine-2,4-diamine
N-{[1-(propan-2-yl)cyclopropyl]methyl}-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-N-(3-methoxyphenyl)piperidine-1-carboxamide
3-({2-[1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[(3-fluoropyridin-2-yl)methyl]-4-(4-methoxyphenyl)-2-methylpiperazine
5-{1-[(2,6-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
1-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
methyl 2-(piperidine-1-sulfonyl)-6-(quinolin-5-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{5-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
1-{1-[(2,5-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(2-methylphenyl)ethyl]-1,3-oxazole-4-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzamide
4-[1-benzyl-5-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2,4-dimethoxy-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine
N-methyl-N-(2-phenylethyl)-5-(piperidin-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(3-{[(1-benzylpyrrolidin-3-yl)carbamoyl]amino}phenyl)-N-methylpropanamide
4-{4-[4-(2-methylpropyl)benzoyl]-2-oxopiperazin-1-yl}benzonitrile
1,5-dimethyl-2-phenyl-4-{[(3-phenylprop-2-yn-1-yl)(propyl)amino]methyl}-2,3-dihydro-1H-pyrazol-3-one
2-(2H-1,3-benzodioxol-5-yl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
N,N-dimethyl-1-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-amine
2-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-1,2-dihydrophthalazin-1-one
1-{2-[1-(2-fluoro-5-methylbenzenesulfonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-[1-(cyclobutylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
6,8-dimethyl-3-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-7-{[(2-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-(3-ethyladamantan-1-yl)-1-(oxolane-2-carbonyl)piperidin-4-amine
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(6-methoxynaphthalen-2-yl)morpholine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-chlorophenyl)methyl]piperidin-3-ol
(1S,5R)-6-propyl-3-[4-(1H-pyrazol-4-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(3-chloro-4-methoxyphenyl)-6-methoxypyrimidin-2-amine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanamide
1-(carbamoylmethyl)-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}morpholin-3-yl)acetic acid
1-[(2-aminopyridin-3-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
2-chloro-N-(1-methyl-5-oxopyrrolidin-3-yl)-5-(trifluoromethyl)benzamide
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl][(2-fluoro-4-methoxyphenyl)methyl]methylamine
1-(2H-1,3-benzodioxole-5-carbonyl)-2-(4-fluorophenyl)piperidine
ethyl (1R,2S)-2-{4-phenyl-1-[3-(pyridin-3-yl)propyl]-1H-imidazol-5-yl}cyclopropane-1-carboxylate
8-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}-N-(1,3,4-thiadiazol-2-yl)benzamide
3-ethoxy-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
5-[(E)-2-cyclohexylethenyl]-4-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3,5-dimethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-ethoxyethyl)-6-(2-methoxyphenyl)pyridazin-3-amine