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5-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carboxamide
2,2,3-trimethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-3-yl]methyl}but-3-enamide
(3aS,6aS)-5-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-[4-(3-hydroxy-3-methylbutyl)benzoyl]-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
N-[(3-methylpyridin-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
4-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-methoxy-4-methylbenzamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
N,N-diethyl-1-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
[2-ethoxy-5-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)phenyl]methanol
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(1R,3S)-3-[({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)carbamoyl]cyclopentane-1-carboxylic acid
1-[2-(4-methoxyphenoxy)ethyl]-4-methylpiperidine
2-(2H-1,3-benzodioxol-5-yl)-N-(1,4-dioxan-2-ylmethyl)acetamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-pentanamidobenzamide
2-cyclopropyl-6-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
1-cyclopropyl-N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-[1-(1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)ethyl]-4-methylpiperazine
1-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
5-methyl-2-[1-(6-methylpyridine-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]pyridine
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(2-methyl-1H-imidazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(3-chlorophenyl)-4-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
3-{5-ethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
1-[benzyl(methyl)amino]-3-[4-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-amino-6-[3-(propan-2-yloxy)phenyl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
1-(2,2-dimethyloxane-4-carbonyl)-4-(2-phenoxyethyl)piperazine
6-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2,4-dimethylpyridine-3-carbonitrile
1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-hydroxypiperidine-4-carboxylic acid
2-{1-benzyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-ethoxyacetyl)-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,6-dimethoxybenzamide
3-[5-(6-cyanopyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-cyclopentylpropanamide
N-[(3S)-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
(1S,5R)-N-(3-cyanophenyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
(1R,2S,9R)-11-{imidazo[1,2-b]pyridazine-3-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
(1R,2R)-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenylcyclopropane-1-carboxamide
3-chloro-5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
8-(cyclopropanesulfonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(hydroxymethyl)-1-(3-methanesulfonylbenzoyl)piperidin-4-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-ol