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N-(4-chloro-3-methoxyphenyl)-2-({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)acetamide
N-benzyl-5-[(4-ethoxypiperidin-1-yl)methyl]pyrimidin-2-amine
1-(4-{2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)propan-1-one
(3aR,6aS)-1-oxo-5-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-[(dimethylamino)methyl]azepan-4-ol
5-ethyl-3-(2-{4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,2,4-oxadiazole
8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{1-[(2,4-dimethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methylpropyl)-1-benzofuran-2-carboxamide
5-{1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)-1-propylpyrrolidin-2-one
4-{4-[(8-methoxyquinolin-2-yl)methyl]piperazin-1-yl}phenol
1-(1-{[2-(furan-2-yl)phenyl]methyl}pyrrolidin-3-yl)-4-methylpiperazine
1-(6-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridin-3-yl)ethan-1-one
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
N-ethyl-1-phenyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]cyclopentane-1-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]acetamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-3-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazole
7-(2-methoxyethyl)-2-{[3-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
3-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indazole
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}furan-2-carboxamide
3-{3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazol-4-yl}pyridine
7-fluoro-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-[(2-chlorophenyl)methyl]-1-(cyclohex-3-en-1-ylmethyl)-1,4-diazepan-5-one
4-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(3-fluorophenyl)piperidine-1-carbonyl]-N,N-dimethylaniline
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
1-[1-(5-fluoro-2-methylbenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
N-({1-[(2-ethylpyrimidin-4-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylfuran-2-carboxamide
(3S,4R)-1-(6-aminopyridine-3-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
[(3-{[1-(3-chlorobenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
N-[(3-chlorophenyl)methyl]-3-[1-(2-phenylethyl)piperidin-4-yl]propanamide
N-{2-[5-(1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}methanesulfonamide
1-methoxy-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
ethyl(oxolan-2-ylmethyl)(piperidin-4-ylmethyl)amine
2-(4-phenylpiperidin-1-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]acetamide
5-ethyl-N-[3-(4-methylpiperazin-1-yl)propyl]pyrimidin-2-amine
N-benzyl{[2-(oxolan-2-ylmethoxy)phenyl]amino}sulfonamide
3-[1-(cyclohexylmethyl)piperidin-3-yl]-N-cyclopropylpropanamide
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-4-fluoro-N-(pyridin-2-ylmethyl)benzamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(5-methylthiophen-2-yl)methyl]amine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-(2-methylphenyl)-3-oxo-3-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propanamide
1-(naphthalen-1-ylmethyl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-{4-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
methyl 6-[(2-methylphenyl)methyl]-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(5-fluoro-2-methoxyphenyl)-1H-indazol-1-yl]acetamide