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4-[5-(2-cyclopentylacetyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
4-[2-(benzyloxy)phenyl]-4H-1,2,4-triazole
2-{2-[(3-cyanopiperidin-1-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}acetamide
5-(methoxymethyl)-N-[4-(5-methyl-4-{[3-(4-methyl-1,3-thiazol-5-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(ethyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
2-(3-acetylphenyl)-N-(propan-2-yl)pyridine-4-carboxamide
3-acetyl-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1H-pyrazole-5-carboxamide
N-methyl-7-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
ethyl 2-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-2-yl}acetate
3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
2,3,5-trimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-3-ethyl-1H-pyrazole-5-carboxamide
4-{5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazole-3-carbonyl}thiomorpholine
N-(2,3-dimethylphenyl)-3-[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]-3-oxopropanamide
4-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
8-(4-propylbenzenesulfonyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
(1S,5R)-6-(5-methylpyrazine-2-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(methylsulfanyl)propyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
1-[(2-methylphenyl)methyl]-3-{[1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]methyl}urea
N,N-bis(propan-2-yl)-2-[3-(pyrrolidin-1-yl)pyrazin-2-yl]benzamide
N-(propan-2-yl)-6-[4-(1H-pyrazol-5-yl)phenyl]pyrimidin-4-amine
2-(2-cyclopropylpyrimidin-5-yl)-7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline
1-(2-chloro-6-methylphenyl)-3-(2-ethyl-2,5-dihydroxypentyl)urea
2-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2,3,4-tetrahydrophthalazine-1,4-dione
dimethyl({[(3S,4R)-1-[4-(methylsulfanyl)benzoyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[3-(furan-2-yl)propyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{5-[3-(cyclopentylcarbamoyl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-[methyl({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amino]-1-phenylethan-1-ol
1-{2-methyl-5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]acetamide
3-(azepane-1-carbonyl)-N-[(5-methylfuran-2-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[ethyl({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]-1λ6-thiolane-1,1-dione
N-methyl-5-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-(1H-imidazol-1-yl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-4-carboxylic acid
4-(1H-imidazol-1-ylmethyl)-N-[3-(2-methylpyrimidin-4-yl)phenyl]piperidine-1-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylbenzamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-benzyl-3-({[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-methyl-8-(6-methylpyrimidin-4-yl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
7-methyl-3-{5-[3-(methylsulfanyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinolin-2-ol
2-({2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-(oxan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-[(4-acetamidophenyl)methyl]-2-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine