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(3aR,6aR)-2-cyclopentyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(4S)-N-(2-chloro-6-methylphenyl)-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
(2S,4S)-4-amino-N-ethyl-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidine-2-carboxamide
3-{[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-{2-[1-(2,5-dichlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
(1R,5S)-6-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-6-azabicyclo[3.2.1]octane
1-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
7-[(3-methoxyphenyl)methyl]-2-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-methoxy-4-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
4-[(1-acetylpiperidin-4-yl)oxy]-N-ethyl-3-methoxy-N-(pyridin-4-ylmethyl)benzamide
1-{2-[methyl(propan-2-yl)amino]acetyl}-4-(2-methylphenoxy)piperidine-4-carboxylic acid
2-[(4-chlorophenyl)methyl]-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methylpropanamide
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxamide
2,3,6-trimethyl-N-(thiolan-3-yl)quinoline-4-carboxamide
6-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-2,3-dimethylquinoxaline
(3S)-1-[3-(3-fluorophenyl)benzoyl]-N,N-dimethylazepan-3-amine
ethyl 4-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}-1H-pyrazole-3-carboxylate
2-(3-chloro-4-hydroxyphenyl)-1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}ethan-1-one
N-cyclopropyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}propanamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
4-(4-fluorophenoxy)-1-(3-methoxypyrazin-2-yl)piperidine-4-carboxylic acid
2-hydroxy-2-methyl-N-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)methyl]propanamide
1-{[1-(4-methoxyphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
5-ethyl-N4,6-dimethyl-N4-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine
4-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-[4-(2-fluorophenyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
2-ethoxy-6-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
3-{[(2-methoxyphenyl)methyl]({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino}propan-1-ol
1-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
7-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(5-methyl-1,2-oxazol-3-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
2-(4-methoxy-2-methylphenyl)-5-methylpyrimidin-4-amine
1-({2-[4-(trifluoromethyl)pyrimidin-2-yl]phenyl}methyl)piperidin-4-one
3-(5-fluoro-2-methoxybenzoyl)-1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidine
4-[(3-methylphenyl)sulfanyl]-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine
3-ethyl-8-[(2-hydroxy-5-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-chloro-2-(propan-2-yloxy)phenyl]methyl}-2-(methylamino)pyrimidine-5-carboxamide
2-(2,5-dimethoxyphenyl)-2-[4-(pyridin-4-ylmethyl)piperazin-1-yl]acetic acid
ethyl 5-(1H-1,3-benzodiazole-5-carbonyl)-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1R,3S)-7-[2-amino-4-(trifluoromethyl)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
2-methyl-N-(oxan-3-ylmethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
6-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1,3-benzothiazole
4-(4-phenyl-1H-pyrazol-5-yl)-1-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]piperidine
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(4-methoxybenzoyl)piperazine
N-tert-butyl-2-methyl-3-[2-(4-methylpiperidin-1-yl)propanamido]benzamide