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8-methoxy-N-[2-(phenylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
5-[3-(propan-2-yloxy)phenyl]pyridin-2-amine
2-(4-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
(1R,7S)-N-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(propan-2-yloxy)propanamide
1-[1-(methylsulfanyl)propan-2-yl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
4-methyl-N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-ol
1-[4-(2-methylphenoxy)piperidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-({4-[(2-fluorophenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}methyl)-N-methylmethanesulfonamide
methyl (1S,3S,3aR,6aS)-3-(3-cyanophenyl)-5-ethyl-1-(hydroxymethyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(1R,5S,6S)-N-(2,3-dihydro-1H-inden-2-yl)-3-[(2-methoxyphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
4-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(thiophene-3-carbonyl)piperidine
3,3-dimethyl-1-({5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-{2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]ethyl}-N-methylmethanesulfonamide
N-[2-(1-hydroxycyclopentyl)ethyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
5-[(3-methoxyphenyl)methyl]-5-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
(2E)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-phenylprop-2-enamide
2-[3-(1H-pyrazol-5-yl)phenyl]-1,3-thiazole
2-({[(2-butoxy-3-methoxyphenyl)methyl]amino}methyl)-6-methyl-3,4-dihydropyrimidin-4-one
(4aR,7aS)-1-(2-methylpropyl)-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-(pent-2-yn-1-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{3-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
1-(1,3-thiazol-2-ylmethyl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
1-(3-chloro-4-methoxyphenyl)-3-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]urea
1-ethyl-4-[4-(4-phenylpyrimidin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
1-(methoxymethyl)-N-{[3-(trifluoromethyl)phenyl]methyl}cyclobutane-1-carboxamide
1-[4-(3-fluorophenyl)phenyl]-N-[(2S)-1-methoxypropan-2-yl]piperidin-4-amine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinoline-6-carbonyl)piperidin-3-yl]propan-1-ol
5-butyl-1'-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-{[(4-methylphenyl)methyl]amino}benzamide
methyl 3-({imidazo[1,2-a]pyridin-2-ylformamido}methyl)-5-[(2E)-3-phenylprop-2-enamido]benzoate
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
1-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(1-methyl-1H-pyrrol-3-yl)-1-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
4-{3-[1-(2-fluoroethyl)-1H-pyrazol-3-yl]phenyl}-2,6-dimethoxypyrimidine
2-amino-6-(2,4-dimethoxyphenyl)-4-(1-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
N-[1-(oxolan-3-ylmethyl)piperidin-4-yl]methanesulfonamide
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(butylsulfanyl)-N4-[(2R)-oxolan-2-ylmethyl]pyrimidine-4,6-diamine
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-ethylpiperazine
3-[1-(9H-fluoren-2-ylmethyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
8-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea