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3-{[(3-hydroxypropyl)amino]methyl}-6,7-dimethoxy-1-[(4-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(3-methylpyridin-2-yl)methyl]acetamide
2-[4-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]pyrimidine
N-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
1-cyclopropyl-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(pyridin-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-({4-[4-(1H-pyrazol-1-yl)phenyl]phenyl}methyl)piperazine
(3S,4R)-3-methoxy-1-(2-phenylquinoline-4-carbonyl)piperidin-4-amine
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
N-benzyl-3-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-methylpropanamide
(1R,5R)-6-(cyclopropylmethyl)-3-(2,3-dihydro-1-benzofuran-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)phenyl]-5-methyl-1,3,4-oxadiazole
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
2-({[2-(2-ethoxyphenoxy)ethyl](methyl)amino}methyl)benzoic acid
7-(4-propylbenzoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-(1H-imidazol-4-yl)-4-phenyl-1-[(4-phenyloxan-4-yl)methyl]-1H-imidazole
(2S,4R)-4-amino-N-ethyl-1-(5-phenoxyfuran-2-carbonyl)pyrrolidine-2-carboxamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
4-cyclopentyl-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylpyrimidin-2-amine
3-(2-amino-1,3-thiazol-4-yl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)propanamide
N,6-dimethyl-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyrimidin-4-amine
N-benzyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
7-[3-(1H-indazol-1-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-{2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
4-[3-(2-phenylethyl)piperidine-1-carbonyl]pyridine
2-methoxy-1-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidin-1-yl)ethan-1-one
1-[(3,4-difluorophenyl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
methyl 1-(2-methoxyethyl)-3-[(1-methylpiperidin-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[(4-methoxynaphthalen-1-yl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(1-methyl-1H-pyrrol-2-yl)-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethane-1,2-dione
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4R)-3-hydroxy-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]pyridine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-fluorophenyl)-N-methyl-3-phenylpropanamide
(4aS,8aR)-1-butyl-6-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-decahydro-1,6-naphthyridin-2-one
1-{[2-(diethylamino)pyridin-3-yl]methyl}-3-(prop-2-en-1-yl)urea
N-(furan-2-ylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
(2S)-N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-hydroxy-3-phenylpropanamide
N-cyclopropyl-3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)benzonitrile
1-(5-fluoro-2-methylbenzoyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
6-[4-(2-methoxyethoxy)phenyl]-N2,N2-dimethylpyrimidine-2,4-diamine
1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-(1-methylpyrrolidin-3-yl)-9-[(2E)-3-phenylprop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
8-acetyl-2-{[4-(carboxymethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl 2-[4-({[2-(1H-imidazol-1-yl)ethyl]carbamoyl}amino)phenyl]acetate
N-[(1-{1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carbonyl}piperidin-4-yl)methyl]acetamide
N4-[2-(4-fluorophenyl)ethyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane