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1-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)pyrrolidin-3-amine
(1R,5R)-3-benzoyl-6-[(3-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
8-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
3-(2,5-dioxoimidazolidin-4-yl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)propanamide
4-[(5-ethylthiophen-2-yl)sulfonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3,5-dimethoxy-2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}benzoic acid
(4aS,8aS)-2-[2-(2-ethylphenoxy)ethyl]-decahydro-2,7-naphthyridin-4a-ol
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
(3aR,6aR)-2-cyclopentyl-5-(pyrimidin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(cyclobutylmethyl)-3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
(3aR,7aS)-5-methyl-2-[4-(1H-pyrazol-1-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(3-fluorophenyl)-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
7-(1,3-benzothiazol-2-yl)-4-{[4-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-9-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
3,5-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}benzamide
9-(cyclopropylmethyl)-1-methyl-4-[(5-propylfuran-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(4-fluorophenyl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
5-(1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
8-(1H-imidazol-2-ylmethyl)-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-3-[1-(3-methylbutyl)-1H-pyrazol-5-yl]-1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]urea
4-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-6-methyl-2-phenylpyrimidine
5-fluoro-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1-(4-methylphenyl)piperazin-2-one
2-(azepan-1-yl)-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
1-[(2,3-difluoro-4-methylphenyl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-benzyl-8-(1-hydroxypropan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-(2-methoxyethyl)-4-(3-methoxypyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
N-[(4-methoxyphenyl)methyl]-3-(2-methyl-1H-imidazol-1-yl)-N-propylpropanamide
5-(3-fluorophenyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,4-triazin-3-amine
{4-[5-(1H-indol-1-ylmethyl)furan-2-carbonyl]-1,4-oxazepan-6-yl}methanol
1-[(3S,4R)-1-[2-(2-methoxy-4-methylphenoxy)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(2R)-2-hydroxy-2-phenyl-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
1-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)piperidin-4-ol
4-chloro-1,5-dimethyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-1H-pyrazole-3-carboxamide
3-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-(3-oxo-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}propyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(3-{3-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenyl}-1H-pyrazol-1-yl)butan-2-ol
1-(6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)azepane
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(naphthalen-1-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-methoxyphenyl)phenyl]-1-(propan-2-yl)piperidine-3-carboxamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-[methyl(naphthalen-1-ylmethyl)amino]azepan-2-one
1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperazine
2-hydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
methyl 6-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyridine-2-carboxylate
1-(4,7-dimethylquinazolin-2-yl)-N-(3-methylbutyl)azepan-4-amine
(2S)-2-amino-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide