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1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[(3-methylpyridin-4-yl)methyl]piperidin-4-amine
ethyl 3-benzyl-1-cyclobutylpiperidine-3-carboxylate
N-{1-[2-(2-oxoazonan-1-yl)acetyl]piperidin-4-yl}methanesulfonamide
2-(hydroxymethyl)-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
1-benzyl-5-(1H-indole-2-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-6-(piperidin-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-4-amine
ethyl 1-(4-methoxyphenyl)-5-{[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-pyrazole-4-carboxylate
3-(piperidin-3-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
(1S)-1-[3-methyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]-2-phenylethan-1-ol
1-[2-methoxy-6-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-(2-methoxy-2-methylpropyl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[1-(4-methylpiperazine-1-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(2S)-1-[2-(2-methoxy-4-methylphenoxy)ethyl]pyrrolidine-2-carboxamide
1-methyl-4-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carbonyl)piperazine-2-carboxylic acid
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
methyl 4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}thiophene-2-carboxylate
7-[2-(methylamino)pyridine-3-carbonyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(1H-pyrazol-1-yl)butanamide
3-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-cyclopropylpropanamide
(2S,4R)-4-amino-N-methyl-1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]pyrrolidine-2-carboxamide
2-{3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
2-({5-[2-(2-hydroxyphenyl)ethyl]-4-methyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-[(2,4-dimethoxyphenyl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
1-(2-methoxyethyl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-6-oxopiperidine-3-carboxamide
1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(pyridin-4-yl)propan-1-one
4-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1-phenylpiperazin-2-one
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-(pyridin-3-yl)propanamide
1-cyclobutanecarbonyl-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]piperidine-4-carboxamide
2-{4-[(morpholine-4-carbonyl)amino]phenyl}-2-(pyrrolidin-1-yl)acetic acid
2-(3-hydroxyphenyl)-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
8-(2,4-dimethylpyrimidine-5-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(dimethylamino)ethyl]-4-(3-methoxypyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxy-4-methylpentan-1-one
N-[4-(methylsulfanyl)phenyl]-6-(pyridine-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
1-ethyl-4-{[({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)amino]methyl}pyrrolidin-2-one
(2R,6R)-11-methoxy-4-methyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
7-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-methyl-4-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,4-dihydroquinoline-2-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(morpholin-4-yl)ethyl]amine
(3R,4S)-4-(3-methoxyphenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-amine
N-[3-(morpholin-4-yl)propyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
(3S,4R)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
1-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
2-methyl-9-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-N,N-diethyl-1-[(3-methylphenyl)methanesulfonyl]pyrrolidine-2-carboxamide