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(3R,4R)-1-(3-chloropyridin-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
3-(methoxymethyl)-1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-(pyridin-2-ylmethyl)-4-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-3-ol
3-{5-[2-(oxan-2-ylmethoxy)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-butoxyacetamide
2-methoxy-1-[1'-(4-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-[1-(2-hydroxy-5-methylbenzoyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-fluoro-N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]benzamide
1-(3-cyano-4-ethoxyphenyl)-3-methyl-3-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
N-[(1-ethylpiperidin-3-yl)methyl]-2-(2-methyl-1H-indol-3-yl)acetamide
N-cyclopropyl-2-[2-(ethylcarbamoyl)phenyl]pyridine-3-carboxamide
2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazole-5-sulfonamide
3-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[(2-methylphenyl)methyl]urea
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(trimethylpyrimidin-4-yl)-decahydroisoquinoline
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][3-(5-methylfuran-2-yl)butyl]amine
4-{[5-(9H-fluoren-9-ylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine
7-(propan-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
2-[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]-2-methylpropanoic acid
3-methyl-8-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-benzyl-8-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
8-(4-hydroxy-2-methylbenzoyl)-1,8-diazaspiro[4.5]decan-2-one
3-(3-hydroxyquinoxalin-2-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
1,1,1-trifluoro-3-{3-[3-(3-methylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
11-{[(2,3-difluorophenyl)methyl]amino}-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
1-[2-(6-hydroxypyrimidin-4-yl)ethyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
4-{2-methyl-3-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]propyl}-4H-1,2,4-triazole
methyl 3-[(2-cyclopentylacetamido)methyl]-5-(furan-2-amido)benzoate
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxybutan-1-one
1-(4-methoxyphenyl)-4-[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]piperazine
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
(1S,6R)-3-methyl-N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
2-(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-({4-methoxy-3-[4-(trifluoromethyl)phenoxy]phenyl}methyl)pyrrolidine
3-methyl-1-[(3-methylphenyl)methyl]-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperazin-2-one
4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
5-{2-[(4-ethylcyclohexyl)formamido]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-methyl-3-(2-{[(piperidin-4-ylmethyl)carbamoyl]amino}phenyl)propanamide
3-cyclopropyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](ethyl)[3-(morpholin-4-yl)propyl]amine
N-(4-{[(prop-2-en-1-yl)carbamoyl]methoxy}phenyl)propanamide
(1r,4r)-4-[({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]cyclohexan-1-ol