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5-{[(4-chlorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(2-ethylpyrimidin-4-yl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
1-[1-(6-cyanopyridin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1-(diethylamino)-3-(2-methoxy-4-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
5-(4-chloro-2-methoxyphenoxymethyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1-hydroxy-2-methylpropan-2-yl)-5-methyl-1H-pyrazole-4-carboxamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-6-(methoxymethyl)-N-methylpyrimidin-4-amine
3-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
5-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
2-(dimethylamino)-4-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidine-5-carboxamide
1-(4-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(2,6-dimethoxy-4-methylphenyl)-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}acetic acid
1-(5-chloropyridin-2-yl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazine
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(2H-1,3-benzodioxol-5-yloxy)ethan-1-one
3-[(3R,4S)-3-(3-cyclopentylpropanamido)-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
2-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
4-[5-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]pyrimidin-2-amine
1-{2-[1-(thiophene-3-sulfonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
methyl 4-({4-[2-(2-chlorophenyl)acetyl]-7-oxo-1,4-diazepan-1-yl}methyl)benzoate
4-[3-cyclopentyl-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
2-[(dimethylcarbamoyl)amino]-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
5-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-4-propylpyrimidine
methyl 4-[2-amino-3-cyano-6-(1H-indol-3-yl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
5-(oxolan-2-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]thiophene-2-carboxamide
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-methyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]urea
6-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]pyridine-3-carboxylic acid
1-methyl-3-{[1-(1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]pyrrolidin-3-yl]acetamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]piperazine
7-propyl-2-[2-(pyrimidin-2-ylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(3-methylpiperidin-1-yl)propanamide
1-[2-methoxy-5-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
N-methyl-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
N-methyl-3-propanamido-N-(quinoxalin-2-ylmethyl)benzamide
1-cyclopropyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
4-(2-hydroxyethyl)-N-[2-(piperidin-1-ylmethyl)phenyl]piperazine-1-carboxamide
3,6-dimethyl-4-[3-(trifluoromethoxy)phenyl]-[1,2]oxazolo[5,4-d]pyrimidine
(5S)-5-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinoline-2-carbonyl}pyrrolidin-2-one
4-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)thiomorpholine
N-[(3S,4R)-1-[2-(2-ethylphenoxy)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-(4-methoxy-3,5-dimethylphenyl)-2-[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]acetic acid
2-({4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-3-methylpyridine
4-{2,7-diazaspiro[4.5]decan-2-ylmethyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N,N-dimethyl-N'-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}butanediamide
2-(2,5-dimethoxyphenyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
2-methyl-N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine