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(3R,4R)-N-cyclohexyl-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carboxamide
3-(3-hydroxybutyl)-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
N-{[(3S,4S)-3-hydroxy-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl]methyl}cyclopentanecarboxamide
2-[(1S,5R)-3-(2-acetylbenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxylic acid
1-methyl-3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
(4aR,8aR)-2-{[4-(prop-2-en-1-yloxy)phenyl]methyl}-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
4-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylacetamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(4-methylbenzenesulfonyl)piperidin-3-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
4-[(4-fluorophenyl)methyl]-1-[4-(methylamino)pyrimidin-2-yl]-3-(propan-2-yl)-1,4-diazepan-5-one
methyl({pyrazolo[1,5-a]pyrimidin-3-ylmethyl})(quinolin-5-ylmethyl)amine
4-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}pyridine
2-methyl-6-(piperidin-4-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidin-4-amine
N,3,6-trimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1-benzofuran-2-carboxamide
N-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
8-(9H-fluoren-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-[(3,4-difluorophenyl)methyl]-2-[5-(methoxymethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decane
1-(2-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl](methyl)amino}pyrimidin-4-yl)pyrrolidin-3-ol
4-{1-[4-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-methylpropan-2-yl}morpholine
3-(4-tert-butylphenyl)-5-(oxolan-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
methyl 4-(3-{[3-(4-fluorophenyl)phenyl]carbamoyl}piperidin-1-yl)-4-oxobutanoate
1-({5-[(2,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
7-(2,3-dimethoxyphenyl)-9-methoxy-4-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-methoxyphenyl)-5-[1-(methylsulfanyl)propan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{2-[4-(6-chloropyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
3-(2-hydroxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
3-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-(1,3-benzothiazol-2-yl)-2-({methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenol
2-{1-[(4-ethoxyphenyl)methyl]-4-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
N,N-dimethyl-5-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}pyridin-2-amine
2-amino-6-(6-methoxynaphthalen-2-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
8-(2,1,3-benzoxadiazol-4-ylmethyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1-(morpholin-4-yl)propan-1-one
(4aS,7aR)-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3-fluoro-2-methylphenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(4aS,8aR)-6-(2,6-dimethoxypyridine-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(4-fluorophenyl)-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]morpholine
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-cyclopropylpropanamide
4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-N-(3-fluorophenyl)-4-oxobutanamide
N-(1-methyl-1H-pyrazol-4-yl)-2-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)acetamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-(2-chlorophenyl)-3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)propanamide
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)pyridazine-4-carboxamide
N,5,7-trimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
5-methyl-4-(1H-pyrazol-1-ylmethyl)-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole