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2-[(3,4,5-trimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane
4-phenoxy-1-[3-(pyrazin-2-yl)propanoyl]piperidine-4-carboxylic acid
5-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
(2S)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
7-(2-hydroxyethyl)-2-(quinoxalin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-phenyl-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-5-yl)phenol
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4,6-dimethylpyridine-3-carbonitrile
N3-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-N5-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-[3-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-N-ethylpyrimidin-2-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
3-ethyl-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-1,2-oxazole-5-carboxamide
(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-[(3-methoxyphenyl)methyl]piperidin-3-yl)methanol
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydroquinoline
2-({[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}amino)-N-(1,3-thiazol-2-yl)acetamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-2-oxo-2-(thiophen-2-yl)acetamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{1,9-dioxaspiro[5.5]undecan-4-yl}acetamide
N-methyl-5-(propan-2-yl)-N-(quinolin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(3S)-1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-N,N-dimethylazepan-3-amine
1-(2-chloro-4-methylphenyl)-3-{[4-(dimethylamino)oxan-4-yl]methyl}urea
6-[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carbonitrile
1-cyclohexyl-4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
(2S,4S)-4-amino-N-methyl-1-[2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetyl]pyrrolidine-2-carboxamide
5,6-dimethoxy-2-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-1,2-dihydroisoquinolin-1-one
3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}-N-[phenyl(pyridin-4-yl)methyl]propanamide
(2S,4R)-1-cyclohexyl-N,N-diethyl-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
8-(6-methoxypyrimidin-4-yl)quinoline
(2S,4R)-1-cyclobutanecarbonyl-N-ethyl-4-(5-ethylthiophene-2-amido)pyrrolidine-2-carboxamide
(2S,4S)-4-(4-{[1-(2,3-difluorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
(2E)-3-(3-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-{[4-(thiophen-2-ylmethoxy)phenyl]methyl}prop-2-enamide
7-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]ethane-1,2-diamine
5-fluoro-1,3-dimethyl-2-[3-(piperidin-1-ylmethyl)piperidine-1-carbonyl]-1H-indole
2-[(3-methoxyphenyl)methyl]-8-[(3-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(cyclopropylmethyl)-5-[1-(2-hydroxyethyl)piperidine-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
8-[2-(ethylamino)pyrimidine-5-carbonyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2-ethoxypyridin-3-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N,N-dimethyl-4-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}aniline
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,5R)-N,N-dimethyl-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[4-({[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}methyl)piperidin-1-yl]-2-methylpropan-1-one
(1S,5R)-6-benzyl-3-{[6-(dimethylamino)pyridin-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-ethoxyethan-1-one
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-3-(1-methyl-1H-pyrazol-5-yl)propanamide
1-methyl-4-(1-phenylcyclopropanecarbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-{1-[(3-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)-N,N-dimethylacetamide
1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
2-methyl-5-{4-[(3-phenyloxolan-3-yl)methyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one