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N-methyl-5-oxo-1-(pyridin-3-ylmethyl)-N-(quinoxalin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}morpholine-2-carboxamide
5-{[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,3-oxazolidin-2-one
5-(4-methylpiperidin-1-yl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
N-(2,2-difluoroethyl)-4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
2-{methyl[5-({methyl[(1-methylpiperidin-2-yl)methyl]amino}methyl)pyrimidin-2-yl]amino}acetic acid
N-[2-(propylsulfanyl)ethyl]thiolan-3-amine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2,3,5,6-tetramethylbenzamide
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(4-phenylmorpholin-2-yl)methyl]acetamide
2-[4-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
4-({3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)quinoline
methyl 6-[(2,3-difluorophenyl)methyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4R)-1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
1-[1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
6-acetamido-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyridine-3-carboxamide
benzyl (7S,9aR)-7-[(4-chlorophenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-[5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
4-acetyl-N-(2-methyl-1-benzofuran-5-yl)-1,4-diazepane-1-carboxamide
3-(2,4-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
1-[4-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)piperidin-1-yl]ethan-1-one
4-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
ethyl 1-(5-methoxyfuran-2-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(prop-2-en-1-yl)acetamide
N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]cycloheptanecarboxamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(2-methylbutyl)piperidine
4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}pyridine-2-carboxamide
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-2-carboxamide
[2-(dimethylamino)ethyl](methyl)(2-{[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]oxy}hex-5-en-1-yl)amine
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
2-(phenylamino)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
methyl (2R)-2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanoate
1-tert-butyl-5-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidine-3-carboxamide
5-ethyl-2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyrimidine
(2S)-2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-2-phenylethan-1-ol
3-(3-methoxypropyl)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
2-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}benzonitrile
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-methyl-4-(propan-2-yl)piperazine-1-carboxamide
N-[4-(2,4-dimethoxypyrimidin-5-yl)phenyl]acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
2-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]-1H-indole
3-ethoxy-4-(prop-2-en-1-yloxy)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
methyl 9-(cyclopentyloxy)-3-(furan-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-methoxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
5-(3-{2-[(4-fluoro-2-methylphenyl)carbamoyl]ethyl}piperidine-1-carbonyl)-2,1,3-benzoxadiazol-1-ium-1-olate
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(isoquinolin-1-yl)-7-azaspiro[3.5]nonan-1-ol
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-5-phenyl-1,2-oxazole