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2-(propylsulfanyl)-5-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}pyrimidine
5-({[(dimethyl-1,3-thiazol-5-yl)methyl](propan-2-yl)amino}methyl)pyrrolidin-2-one
3-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-N,N-dimethylaniline
N-(1-methoxypropan-2-yl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-4-(piperidin-3-yl)benzamide
4-[(4-ethylphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(5-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
N-cyclopentyl-N-({4-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)furan-2-carboxamide
2,6-difluoro-N-(1-phenylbutyl)benzamide
5-(4-methyl-1,4-diazepan-1-yl)-2-(pyrrolidin-3-ylmethyl)-2,3-dihydropyridazin-3-one
4-{3-[3-(pyridin-3-ylmethyl)piperidin-1-yl]propanamido}benzamide
N-methyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-N-(2-phenylethyl)piperidin-3-amine
1-[2-(dimethylamino)ethyl]-5-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-3-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}thiophene-3-carboxamide
(5-{[2-(4-methoxy-3-methylphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}furan-2-yl)methanol
2-[(4-ethoxyphenyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
1-cycloheptyl-6-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide
N,4-dimethyl-1-{4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-6-yl}piperidine-4-carboxamide
(2S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-methyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
3-(2-{2-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-oxazolidin-2-one
1-[(2,3-dimethoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperazine
5-methyl-1-[4-(4-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
ethyl 2-{4-[4-(dimethylcarbamoyl)-8-methylquinolin-2-yl]-1H-pyrazol-1-yl}acetate
1-(1,4-dioxan-2-ylmethyl)-3-[4-(furan-2-yl)phenyl]-1-methylurea
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
5-(4-methoxyphenyl)-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1,2,4-triazin-3-amine
methyl 4-(4-{[4-(2-fluorophenoxy)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-1,4-diazepane
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
2-cycloheptyl-1-(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-(prop-2-en-1-yl)-5-[4-(pyridin-4-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
{[(3S,4R)-1-(4,6-dimethoxypyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
1-[(4-methylphenyl)amino]-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]cyclopentane-1-carboxamide
[(1-benzylpyrrolidin-3-yl)methyl](1H-imidazol-2-ylmethyl)methylamine
5-{1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-phenyl-1H-imidazol-5-yl}-2-(propan-2-yl)pyrimidine
(1S,5R)-6-benzyl-3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
({5-[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
6-amino-N-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}pyridine-2-carboxamide
5-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1,3-benzothiazol-2-amine
4-ethyl-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[4-({1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
N-(3-hydroxy-3-phenylpropyl)-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(pyridin-4-yl)propanamide
(3S,4R)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
2-ethoxy-5-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}pyridine
N-[3-(difluoromethoxy)phenyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide