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5-propyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-oxazole-3-carboxamide
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(cyclohexylmethyl)piperidin-2-one
N,N-dimethyl-2-{9-oxo-1-oxa-8-azaspiro[4.6]undecan-8-yl}acetamide
{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)(3-methylbutan-2-yl)amine
4-{[3-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]methyl}morpholine
4-methyl-N-{3-[2-(morpholin-2-yl)acetamido]phenyl}benzamide
3-{[7-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
2-(2-{[1-(3,5-dimethylphenyl)piperidin-4-yl]amino}ethyl)-1,2-dihydrophthalazin-1-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N,N-bis(prop-2-en-1-yl)propanamide
1-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
5-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
(3R,4R)-1-[1-(3,5-dimethylphenyl)piperidin-4-yl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
6,8-dimethyl-4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-2H-chromen-2-one
4-ethyl-1-[2-(naphthalen-1-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[3-(3-methylphenyl)phenyl]piperidin-4-yl}piperidine-4-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,N-dimethylazepan-4-amine
2-[5-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
1-({[1-(dimethyl-1,3-thiazol-2-yl)propyl]carbamoyl}methyl)piperidine-4-carboxamide
4-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-N-methyl-1,3-thiazol-2-amine
3-(2,3-dihydro-1H-inden-2-yl)-8-(furan-3-ylmethyl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(5-methylfuran-2-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
6-chloro-8-methyl-4-[3-(pyridin-4-yl)azetidin-1-yl]quinoline
1-[4-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)phenyl]imidazolidine-2,4-dione
N-methyl-N-({5-[4-phenyl-1-(prop-2-en-1-yl)-1H-imidazol-5-yl]furan-2-yl}methyl)methanesulfonamide
(3R,4S)-1-(1-benzyl-1H-pyrazole-4-carbonyl)-4-phenylpyrrolidin-3-amine
N4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N4-methyl-6-(propan-2-yloxy)pyrimidine-2,4-diamine
8-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
2,5-dimethyl-3-{4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl}pyrazine
9-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
N-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidine
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-{[(2-methoxy-2-methylpropyl)amino]methyl}-1,2-dihydroquinolin-2-one
3-{6-[(dimethylamino)methyl]-1,4-oxazepane-4-carbonyl}-2-methylphenol
2,6-difluoro-4-methoxy-N-methyl-N-(quinolin-6-ylmethyl)benzamide
4-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}piperazine-1-carboxamide
[(3R,4R)-1-[(2-chloro-3,6-difluorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(6-ethyl-2-methylpyrimidin-4-yl)-N-methylpiperidin-3-amine
2-(2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(3R,5S)-1-benzyl-N-cyclopentyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-3-carboxamide
3-(3-methoxypyrrolidine-1-carbonyl)-N-[2-(pyrrolidin-1-yl)ethyl]benzene-1-sulfonamide
ethyl 5-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
6-methyl-2-(4-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-[4-(6-hydroxy-1,4-diazepane-1-carbonyl)phenyl]imidazolidine-2,4-dione
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide