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1-{3-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[2-(4-chlorophenyl)ethyl]-2-[2-(pyridin-3-yl)piperidin-1-yl]acetamide
(2S)-1-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-3-hydroxy-2-(methylamino)propan-1-one
N-[4-({1-ethyl-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)phenyl]acetamide
5-methoxy-2-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-4H-pyran-4-one
5-(4-fluorophenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-{3-[3-(4-methylphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N3-{2-[3-(propan-2-yloxy)phenyl]ethyl}piperidine-1,3-dicarboxamide
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
8-[5-(azepane-1-carbonyl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]quinoline
N-[(5-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-methylpiperazin-1-yl)-2-methoxyethan-1-one
4-(5-methoxy-1H-indole-2-carbonyl)-1,4-oxazepan-6-ol
(1R,5R)-6-(cyclobutylmethyl)-3-(2-methyl-5-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
methyl (2S,4R)-4-hydroxy-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidine-2-carboxylate
1-(4-methoxyphenyl)-2,2-dimethyl-4-(2-methyloxane-2-carbonyl)piperazine
1-(2-{1-[(2,3-difluoro-4-methoxyphenyl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
(2S,4R)-4-amino-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
N-(5-cyano-1,3-thiazol-2-yl)-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)benzamide
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-(3-chlorobenzoyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
1-cyclopentyl-4-({[(4-methanesulfonylphenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
N-[(2-aminopyrimidin-5-yl)methyl]-1-cyclopentanecarbonyl-N-methylpiperidine-4-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-methyloxane-2-carboxamide
1-(piperidin-3-yl)-3-(1,3,4-thiadiazol-2-yl)urea
methyl (2S,4S)-4-(2,3-dimethyl-1H-indole-5-amido)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
N-benzyl-1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
3-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,4,4-trifluorobutanamide
3-{[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({5-[(4-ethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
4-(benzyloxy)-1-(thiophene-3-carbonyl)piperidine
1-cycloheptanecarbonyl-N-(4-fluorophenyl)piperidin-3-amine
7-(2-methoxyethyl)-2-[3-(pyrazin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-[2,6-dimethyl-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-benzyl-3-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}oxy)benzamide
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2-methoxyphenol
1-{2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}cyclopentan-1-ol
2-[(4-chlorophenyl)methyl]-N-[1-(pyridin-4-yl)propyl]-1,3-benzoxazole-5-carboxamide
1-methyl-3-(naphthalen-2-ylmethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1s,4s)-N1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}cyclohexane-1,4-diamine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(oxolane-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one