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3-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
7-(4-chloro-2-hydroxybenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aR,7aS)-4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3,5,7-trimethyl-N-(2-methylpropyl)-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
methyl 4-[6-amino-5-cyano-4-(4-hydroxy-3-methylphenyl)pyridin-2-yl]-5-methylfuran-2-carboxylate
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
N-{[1-(1H-indol-2-ylmethyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
1-(4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
(4aR,7aS)-1-cyclobutanecarbonyl-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-fluoro-4-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methylphenyl)methyl]acetamide
N,N-diethyl-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
3-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)benzamide
2-(dimethylamino)-2-(2-methylphenyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
methyl 6-[(1-methyl-1H-indol-3-yl)methyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3-methylbutyl)-8-(1-methylpiperidine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}morpholin-2-yl)ethan-1-ol
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(pyridin-4-yl)-1H-pyrazol-1-yl]acetamide
2-(2-aminoethyl)-N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]quinazolin-4-amine
ethyl 4-[(4-chlorophenyl)methyl]-1-[2-(cyclohex-1-en-1-yl)acetyl]piperidine-4-carboxylate
2-[4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-cyclopropyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
(2R,3R,6R)-5-(2-ethylpyridine-4-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)thiophene-2-carboxamide
N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-propyl-1,2-oxazole-3-carboxamide
N-(1-benzylpyrrolidin-3-yl)-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
ethyl 3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
(3aR,6aR)-2-methanesulfonyl-N,N-dipropyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl 2-[3-(2,6-dimethylphenoxy)azetidin-1-yl]pyridine-3-carboxylate
2-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1,3-thiazole
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-methanesulfonamidopropanamide
(2S,4S)-N-[2-(4-fluorophenyl)ethyl]-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
2-amino-2-methyl-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
5-cyclopropyl-N-[(2-ethoxypyridin-3-yl)methyl]-1,3,4-oxadiazol-2-amine
1-[(2-chlorophenyl)methyl]-N-methyl-N-[3-(pyrrolidin-1-yl)butyl]-1H-1,2,3-triazole-4-carboxamide
N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-1-benzofuran-3-carboxamide
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(3-methylpyridin-2-yl)ethyl]benzamide
6-{3-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(1-methylcyclopropyl)-N-(oxolan-2-ylmethyl)propanamide
8-(8-chloroquinolin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
2-methyl-5-{3-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]phenyl}-1,3,4-thiadiazole
1-(6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridin-3-yl)ethan-1-one
1-[(3-hydroxy-4-methoxyphenyl)methyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
5-({[(3R,5S)-1-benzyl-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-yl]amino}methyl)-2-methoxyphenol