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N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pyridin-4-ylmethyl)oxane-4-carboxamide
7-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-oxa-7-azaspiro[4.5]decane
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]urea
1-[1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
8-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]quinoline-7-carboxamide
1-{[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(1H-indol-6-ylmethyl)-5-oxopyrrolidine-3-carboxylic acid
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(1,3-thiazol-4-ylmethyl)piperidin-4-ol
5-chloro-6-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]pyridine-3-carboxylic acid
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
N-{4-[(furan-2-ylmethyl)(prop-2-yn-1-yl)carbamoyl]phenyl}-2-methylfuran-3-carboxamide
7,7-dimethyl-2-(5-methyl-1H-pyrazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(1-{1,9-dioxaspiro[5.5]undecan-4-yl}piperidin-4-yl)pyridine
1-cyclopentyl-N-methyl-6-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
2-(1H-imidazol-2-yl)-N-[1-(4-methanesulfonylphenyl)ethyl]benzamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenoxyethyl)acetamide
(3aS,6aS)-2-pentyl-5-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[({1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
1-[(3-methoxyphenyl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-cyano-5-fluorobenzamide
3-methyl-7-[(4-phenoxyphenyl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2-hydroxyethyl)-6-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]imidazo[1,2-a]pyridine-2-carboxamide
2-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-3,5,7-trimethyl-1H-indole
N-cyclopropyl-2-(2,5-dioxoimidazolidin-1-yl)-N-(1H-indol-5-ylmethyl)acetamide
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
3-[1-(7-methyl-1-benzofuran-2-yl)-N-(2-phenylethyl)formamido]propanamide
2-fluoro-5-sulfamoyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1-methyl-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-{5-[5-(oxolan-2-yl)thiophen-2-yl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
5-methyl-3-[2-(morpholin-4-yl)ethyl]-5-{1-[2-(naphthalen-1-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(4-cyclohexylpiperazine-1-carbonyl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
5-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}-2-(furan-2-yl)pyrimidine
ethyl 3-[(2-fluorophenyl)methyl]-1-[2-(furan-2-yl)-2-oxoacetyl]piperidine-3-carboxylate
N-methyl-6-oxo-1-(2-phenylethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{4-[(3-hydroxy-2,2-dimethylpropyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-[4-(4H-1,2,4-triazol-4-yl)phenyl]pentanamide
N-{1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(1S,5R)-3-(5-methylpyrazine-2-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
8-(2,5-dimethylfuran-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-3-methyl-5-propyl-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)acetamide
N-[1-(7-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-methoxypropanamide