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4-{3-[5-(2-methyl-1,3-thiazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2,3-dihydro-1-benzofuran-2-carboxamide
2-{3-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
1-benzyl-1',5',6',7'-tetrahydrospiro[azepane-4,4'-imidazo[4,5-c]pyridine]-7-one
4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
3-(2-methylphenyl)-1-(2,3,6-trimethylquinoline-4-carbonyl)pyrrolidin-3-ol
2-(2-{methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N2-tert-butyl-6-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N4-(2-methylphenyl)-1,3,5-triazine-2,4-diamine
2-(2-benzyl-3-oxopiperazin-1-yl)-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
methyl 2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-phenylacetate
2-{5-[(5-acetylthiophen-3-yl)methyl]-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-{2-[5-(pyrrolidine-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}prop-2-en-1-one
4-methyl-2-{2-oxo-2-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
N-(3-{4-[(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}phenyl)-4-phenylbutanamide
9-(2-hydroxy-4-methylpentanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-ethanesulfonamidobenzoyl)-3-propylpiperidine-3-carboxylic acid
N-({1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl}methyl)-4-fluorobenzamide
N-[(3-methylphenyl)methyl]-3-(2-oxoimidazolidin-1-yl)-N-(propan-2-yl)benzamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)pyridine-2-carboxamide
4-({5-[1-(furan-2-ylmethyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
benzyl[(5-ethylpyridin-2-yl)methyl](1,3-thiazol-2-ylmethyl)amine
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-{[3-(pyrrolidin-1-yl)phenyl]methyl}urea
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
(4aS,7aR)-1-(2,6-difluoro-3-methylbenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-[(3-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(pyridin-2-yl)acetamide
N-(2-methyl-1H-1,3-benzodiazol-6-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
3-fluoro-N-[(2R,3R)-2-methoxy-1'-(thiophen-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
(3R,4S)-4-[4-(2,8-dimethylquinoline-4-carbonyl)-1,4-diazepan-1-yl]oxolan-3-ol
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl]pyridine-2-carboxamide
(1S,5R)-3-[3-(morpholin-4-yl)propanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2,3-dihydro-1H-inden-1-yl)-N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)acetamide
2-ethoxy-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-one
N,2-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-hydroxy-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-2-carboxamide
2,7-dioxo-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1,3-diazepane-4-carboxamide
9-[(3,5-difluorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-butylpyrrolidin-1-yl)-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-amino-6,8-dimethyl-4-(6-methyl-1H-indol-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
1-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
(1S,5R)-6-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
4-({[7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)-1,3-thiazol-2-amine
3-(2-methoxyphenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
3-(8-methoxy-2-methylquinolin-5-yl)pyrazine-2-carbonitrile
(2S,4S)-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide