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1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-fluoro-2-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
1-(4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}phenyl)imidazolidine-2,4-dione
1-cyclopropyl-5-oxo-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
1-(2-fluorophenyl)-N-(1,3-thiazol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
8-[2-(1H-pyrrol-1-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
1-[(4-fluorophenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4-diazepane
1-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
2-(2-methoxypyrimidine-5-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
3-[2-(dimethylamino)ethyl]-8-[3-(5-methylfuran-2-yl)butyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[2-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-imidazol-1-yl]-N,N-dimethylethane-1-sulfonamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,2-bis(prop-2-en-1-yl)piperidine
methyl (2R,4S)-1-[(2E,4E)-5-(4-chlorophenyl)penta-2,4-dien-1-yl]-4-hydroxypiperidine-2-carboxylate
ethyl 1-[(2,5-dimethylthiophen-3-yl)sulfonyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}-6-methoxyphenol
[(3,5-dimethoxyphenyl)methyl]({[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl})amine
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}propanamide
(1S,5R)-3-(quinolin-6-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1-propyl-1H-imidazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)piperazine
1-cyclopropyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrrole-2-carboxamide
7-cyclohexyl-2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2,7-diazaspiro[4.5]decan-6-one
N-(2,3-dihydroxypropyl)-N'-(2,4-dimethoxyphenyl)-N-methylpropanediamide
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-methylpyridine-4-carboxamide
(2S,4R)-N-ethyl-4-(2-hydroxyacetamido)-1-[3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carboxamide
N'-(2H-1,3-benzodioxol-5-ylmethyl)-N'-(pyridin-3-ylmethyl)-N-(1,3,4-thiadiazol-2-yl)ethanediamide
3-cyclopentyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
1-ethyl-6-oxo-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
N-[(2R,4S,6R)-2-cyclohexyl-6-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]oxan-4-yl]acetamide
6-methoxy-N,3-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-benzofuran-2-carboxamide
3-(4-{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)propanamide
[2-(2,6-dimethylphenoxy)ethyl](ethyl)[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]amine
5-methoxy-1,2-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1H-indole-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
6-methyl-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-{2-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]ethyl}-1,3-oxazinan-2-one
6-{[(3-methylphenyl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
6-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
5-(methoxymethyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}furan-2-carboxamide
2-(2,5-dimethylfuran-3-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-({4-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperazin-1-yl}methyl)benzonitrile
N-(1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methyl-3-(methylsulfanyl)propanamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-(morpholin-3-yl)ethan-1-one
4-[(2-methylphenyl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one