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1-(2-methylpyridin-4-yl)-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,4-diazepane
1-{2-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
3-chloro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
2-ethyl-6-[4-(4-methylphenyl)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-phenoxy-N-[1-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
4-ethyl-1-methyl-3-{1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R)-1-[(1-{[1-(3-methylpyrazin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-ol
2-benzyl-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
1'-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-3-yl)oxy]methyl}pyridine
4-benzyl-3-ethyl-1-(pyridine-3-sulfonyl)-1,4-diazepan-5-one
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-(furan-3-ylmethyl)-N-methylacetamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1-(6-methylpyrimidin-4-yl)piperidin-4-amine
N-(oxolan-3-yl)-6-phenylpyridazin-3-amine
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
3-(1-methyl-1H-1,3-benzodiazol-5-yl)-1-{[3-(pyrrolidin-1-yl)phenyl]methyl}urea
1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
ethyl 1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(4-hydroxypiperidin-1-yl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}acetamide
1-{1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}piperidin-4-ol
2-({[1-(hydroxymethyl)cyclobutyl]methyl}sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
3-[5-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(2-ethylbutyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N,1-dimethyl-N-(quinolin-5-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)amine
1-methyl-5-(3-methyl-3-phenylpiperidine-1-carbonyl)-1,2-dihydropyridin-2-one
2-fluoro-N-methyl-N-[3-(oxolan-2-yl)propyl]-5-sulfamoylbenzamide
N-methyl-7-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
(3S,5R)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
4-{1-[2-(2-chlorophenyl)ethyl]-1H-imidazol-2-yl}-1-methylpiperidine
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(2-methoxyphenyl)piperazine
3-(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
(3R,4R)-1-(4-cyclopentylpyrimidin-2-yl)-4-(morpholin-4-yl)piperidin-3-ol
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N-[(4-methoxyphenyl)methyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(thiophene-3-sulfonyl)piperidine
(1S,5R)-3-[(2-butyl-1H-imidazol-4-yl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
7-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-methoxypyrazine
1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-N,N-diethylpyrrolidin-3-amine
(1S,5R)-6-(2-methoxyethyl)-3-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(propan-2-yl)propanamide
(1-{[1-(4-methylpyridin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetic acid
N-[2-(pyridin-2-ylsulfanyl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide