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3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(thiophene-3-carbonyl)piperidin-4-yl]oxy}benzamide
4-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-2,6-dimethylphenyl acetate
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,3R)-3-amino-1'-(5-methyl-1H-indazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
1-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}piperidine
N-{[4-(4,4-difluoropiperidine-1-carbonyl)phenyl]methyl}-4-methylaniline
5-acetyl-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,4-dimethyl-1H-pyrrole-3-carboxamide
(1R,2S,4R)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide
ethyl 4-(2-methoxyethyl)-1-[4-(4-methoxyphenyl)butan-2-yl]piperidine-4-carboxylate
1-(2-methoxyethyl)-3-(2-methylphenyl)-3-{2-oxo-2-[3-(2-phenylacetyl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
1-(4-fluorophenyl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}methanesulfonamide
N-[2-(5-methylfuran-2-yl)ethyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(3R,4S)-3,4-dimethyl-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-4-ol
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
ethyl 4-(2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazine-1-carboxylate
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-cycloheptyl-N-[2-(methylsulfanyl)ethyl]-6-oxopiperidine-3-carboxamide
ethyl 4-(cyclopropylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-1,4-oxazepan-5-one
N-benzyl-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-phenyl-4-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
2-(piperidine-1-carbonyl)-3-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrazine
N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
6-(2-chlorophenyl)-N,7-bis(cyclopropylmethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[5-(oxane-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazole
1-benzyl-N3-[1-(furan-2-yl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-ethyl-2-(1H-imidazol-1-yl)-N-[1-(4-methoxyphenyl)propyl]acetamide
(benzylsulfamoyl)[2-(methylsulfamoyl)ethyl]amine
1-[2-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)ethyl]piperidine
2-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4-fluorophenyl)-2,2-dimethyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]cyclopropane-1-carboxamide
4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
[1-(2-methyl-1H-imidazol-1-yl)propan-2-yl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-(3-hydroxypropyl)-8-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-tert-butyl-N-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidine-3-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2,1,3-benzoxadiazole
1-[(2-ethoxyphenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[2-(methylsulfanyl)ethyl]-1,2-oxazole-3-carboxamide
4-[2-(methylsulfanyl)phenyl]-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[5-(cyclopropylcarbamoyl)-2-methoxyphenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
N-(2-methoxyethyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
N,N-diethyl-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
dimethyl[2-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)ethyl]amine
(1S,3R)-N1-[2-(2,5-dimethylphenoxy)ethyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
7-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine