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1-methyl-8-[2-(methylamino)pyridine-4-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-ethyl-6-(2-fluoro-4-methoxyphenyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl 3-[(2,3-dihydro-1-benzofuran-2-ylformamido)methyl]-5-(2-phenylacetamido)benzoate
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)oxan-4-amine
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-methoxypyridine
N-(2-methoxyethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(2-methoxyethyl)-N-(propan-2-yl)propanamide
2-[1-(cyclohexylmethyl)-4-[1-(2-fluorophenyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-(3-methoxypropyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-methyl-1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]azetidin-3-yl}piperidine
1-[6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]-4-phenylazepane
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N-benzyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-5-methyl-1H-indole-2-carboxylic acid
6-ethyl-1-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[2-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
2,7,8-trimethyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]quinoline-4-carboxamide
1-[2-(morpholin-4-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(4R)-N,3-dimethyl-N-(quinolin-5-ylmethyl)-1,3-thiazolidine-4-carboxamide
N-(propan-2-yl)-3-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propanamide
N-[2-chloro-5-(piperidine-1-carbonyl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
3-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
(1R,3s,6r,8S)-4-[(4-methyl-1H-imidazol-2-yl)methyl]-4-azatricyclo[4.3.1.13,8]undecane
1-(2-ethoxyethyl)-N-[2-(5-methylthiophen-2-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(1-methyl-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
1-(cyclopropylmethyl)-4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
3-(1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-[(3R,4S)-1-(3-chloro-4-ethoxybenzoyl)-4-cyclopropylpyrrolidin-3-yl]acetamide
2-(3-chlorophenoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
3-phenyl-6-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyridazine
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-methyl-4-[2-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)ethyl]piperidin-4-ol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
3-(4-methylphenoxymethyl)-1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]piperidine
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-methoxyethan-1-one
3-(1H-imidazol-1-ylmethyl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-(2-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
1-[7-(cyclohexylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-phenylethane-1,2-dione
methyl 4-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)benzoate
5-{[benzyl(methyl)amino]methyl}-N-[2-(thiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(carbamoylmethyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}piperidine-4-carboxamide
3-[(2R,3R,6R)-5-(1,4-dithiepan-6-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
8-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-tert-butyl-N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide