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N-benzyl-5-[3-(diethylamino)pyrrolidine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-methyl-9-[2-(1H-pyrazol-1-yl)butanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,6R)-3-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
N-[3-(4-fluorophenyl)phenyl]-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidine-3-carboxamide
6-[(3,5-dimethoxyphenyl)methoxy]-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1-(propan-2-yl)-1,4-diazepan-2-one
1-(1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-(trifluoromethyl)benzamide
5-(furan-3-yl)-1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-[(4-methylphenyl)methyl]piperazin-2-one
4-ethyl-1-[(3S)-3-hydroxy-3-phenylpropyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-[3-(propan-2-yloxy)propyl]piperidine-4-carboxamide
1-(5-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
N-cyclopentyl-3-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
7-chloro-4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]quinoline
N-(2-hydroxyethyl)-N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyridin-4-yl)propyl]pyridin-2-amine
1'-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}spiro[indene-1,4'-piperidine]
5-methoxy-2-{[3-(4-phenylbenzoyl)piperidin-1-yl]methyl}pyridin-4-ol
N-[3-(2-methoxyphenyl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-[6-(4-fluorophenyl)pyridazin-3-yl]pyridin-3-amine
1-{3-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}pyrrolidin-2-one
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
N-(3-hydroxy-2,2-dimethylpropyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(pyridine-3-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1,4-dimethylpiperidin-4-yl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperidine-4-carbonitrile
N-[2-(2,4-difluorophenyl)-1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
4-(1-ethenyl-1H-pyrazol-4-yl)-3-(4-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]-2H-chromene-3-carboxamide
7-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]-2-amino-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-[3-(2-cyclopentylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methoxypyrimidine
5-{[2-(methoxymethyl)piperidin-1-yl]methyl}-8-methylquinoline
N-methyl-1-(oxolane-2-carbonyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-3-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]propanamide
2-(4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
5-(2-fluorophenyl)-N-[2-(propane-2-sulfonyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-({[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenol
N-(3-chloro-2-methylphenyl)-2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-4-fluorobenzene-1-sulfonamide
3-benzyl-5-[(2,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazole
2,6-dimethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
4,6-dimethyl-3-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-1,2-dihydropyridin-2-one
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one
10-methoxy-5-(5-propyl-1,2-oxazole-3-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-cyclopentyl-1-[4-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
1-(oxolan-3-ylmethyl)-4-(3-phenylpropyl)-1,4-diazepane