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N-[2-(diethylamino)ethyl]-9-(3,4-difluorophenyl)-15-methyl-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
1-{4-[(cyclooctylamino)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(4-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}phenyl)cyclobutanecarboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}thiophene-3-carboxamide
3-benzyl-8-(1-hydroxypropan-2-yl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(1H-1,2,4-triazol-1-yl)butanamide
2-amino-4-[3-(morpholin-4-ylmethyl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
3-cyclohexyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methoxyphenoxy)piperidine
(2R,6R)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
N-{3-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}acetamide
N-cyclopropyl-4-methoxy-3-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
dimethyl({4-[(2-methylnaphthalen-1-yl)methyl]-1,4-oxazepan-6-yl}methyl)amine
N-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-4-(pyridin-4-yl)piperazine-1-carboxamide
9-methoxy-N-methyl-3-(6-methylpyridine-2-carbonyl)-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-3-propanamidobenzamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(propylsulfanyl)ethan-1-one
9-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-[(4-fluoro-3-methoxyphenyl)methyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-(trifluoromethyl)morpholine
1-{[5-(1-benzoylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}azepane
6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-N-(propan-2-yl)pyrimidin-4-amine
3-(naphthalene-1-carbonyl)-1-[2-(1H-pyrazol-4-yl)ethyl]piperidine
6-(2,5-dimethylfuran-3-yl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methylpropanamide
N-[(5-chloro-1H-indol-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
7-(2-methoxyphenyl)-2-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1S,6R)-9-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-cyclopropyl-1-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propan-1-one
1-ethyl-N-[(3-methoxyphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2,3-dihydro-1H-inden-1-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)azepan-4-amine
6-({[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}amino)-2-methylheptan-2-ol
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-5-methylimidazo[1,2-a]pyridine-2-carboxamide
(3aR,6aS)-5-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}ethane-1-sulfonamide
1-(4-fluorophenyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopropane-1-carboxamide
(3S)-4-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-3-ethylmorpholine
N,N-dimethyl-2-[(1S,5R)-3-[2-(methylsulfanyl)pyridine-3-carbonyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(3,5-dimethyl-4-phenyl-1H-pyrazol-1-yl)-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
pyridin-2-yl[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]methanol
(3aS,6aS)-2-(2-methoxyethyl)-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
phenyl (7S,9aR)-6,9-dioxo-7-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidin-2-one