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3-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[3-methoxy-5-(trifluoromethyl)phenyl]urea
2-(ethoxymethyl)-N-(1H-imidazol-2-ylmethyl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
2-(3-methoxypropyl)-9-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2,3-dimethylquinoxaline-6-carboxamide
1-(5-chloro-2-methylphenyl)-4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
2-[2-(1H-imidazol-1-yl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(4-methylphenoxy)acetyl]piperidin-3-yl}propanamide
(1R,5S,8S)-8-methoxy-3-({3-[3-(morpholin-4-yl)propoxy]phenyl}methyl)-3-azabicyclo[3.2.1]octane
5-(2-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(4-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperazin-1-yl)propan-1-ol
1-(4-ethoxybenzoyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-5-cyclopropyl-1,3,4-oxadiazol-2-amine
cyclopentyl 4-[({[4-(hydroxymethyl)oxan-4-yl]methyl}carbamoyl)amino]benzoate
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(3-methylphenyl)piperazine
(3R,4R)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-3,4-dimethylpyrrolidin-3-ol
2-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-4H-chromen-4-one
1-[6-(3,4-dichlorophenyl)pyridin-2-yl]piperazine
N-{1-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
methyl 3-(cyclobutylmethoxy)-5-{[(5-methyl-1H-pyrazol-3-yl)methyl]carbamoyl}benzoate
2,5,7-trimethyl-N-[(1-methylpyrrolidin-3-yl)methyl]quinoline-4-carboxamide
N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}pyrrolidine-2-carboxamide
1-(4-methoxyphenyl)-4-(6-methylpyridine-2-carbonyl)piperazin-2-one
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-propylpiperazine
4-{4-[(4-ethoxypiperidin-1-yl)methyl]phenyl}-2-methylbutan-2-ol
7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-4-(quinoline-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-({1-[(1-ethyl-1H-indol-6-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
methyl 7-oxo-3-[2-(phenylsulfanyl)acetyl]-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[4-fluoro-3-(2-methylpropanamido)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-5-phenyl-1H-pyrazole-3-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
N-cyclopentyl-3-[(1,4-dioxan-2-ylmethyl)(methyl)sulfamoyl]benzamide
5-methoxy-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidine
2-ethoxy-5-(2-{[(3R,4R)-4-hydroxypyrrolidin-3-yl]amino}pyrimidin-4-yl)benzoic acid
3-(aminomethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)acetamide
1-(2-aminopyrimidin-4-yl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
N-(2-benzamido-5-methylphenyl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
8-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[2-(benzenesulfonyl)ethyl]-3-(4-chlorobenzoyl)piperidine
N-ethyl-1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidine-3-carboxamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1H-pyrazole-3-carboxamide
2-{2-[1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[(4-methoxyphenyl)methyl]-2-(morpholin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
4-(benzyloxy)-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine
4-[(3R,5R)-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidine-3-carbonyl]morpholine
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide