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1-(1-oxo-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-2-yl)pyrrolidin-2-one
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-(4-hydroxyphenyl)-2-phenylpropanamide
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(pyridine-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
2-methyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-1,3-thiazole-4-carboxamide
5-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
7-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
ethyl 1-[(2-ethoxy-2-oxoethyl)carbamoyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
(2S)-3-hydroxy-2-[3-(3-hydroxyquinoxalin-2-yl)propanamido]propanamide
4-(cyclopropylmethyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-[2-(4-methoxyphenyl)ethyl]-N-[2-(2-methylphenyl)ethyl]-6-oxopiperidine-3-carboxamide
(3S,4R)-3-methoxy-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-6-[(2-methylpyrrolidin-1-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S)-1-({3-[4-(piperidin-1-yl)butoxy]phenyl}methyl)pyrrolidin-3-amine
4-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-methoxypyridine-3-carbonitrile
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[(2,6-difluorophenyl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,5R)-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 2-[1-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)piperidin-2-yl]acetate
N-(cyclopropylmethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-propylpropanamide
5-[(4-methyl-1H-imidazol-1-yl)methyl]-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
2-(4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
2-(2-hydroxyethyl)-8-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(1-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(3-methoxybenzoyl)piperazine
1-(3-propyl-1H-pyrazole-5-carbonyl)azetidine-3-carboxylic acid
6-{4-[(8-methylquinolin-5-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
(2E)-N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-3-(thiophen-2-yl)prop-2-enamide
4-(2-ethylpyrimidine-5-carbonyl)-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
methyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[3-(trifluoromethyl)phenyl]methyl}amine
3-{1-[(3,5-dimethylphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
(2S,4S)-4-amino-N-ethyl-1-[2-hydroxy-3,5-bis(propan-2-yl)benzoyl]pyrrolidine-2-carboxamide
N-methyl-3-[N-methyl-1-(3,4,7-trimethyl-1H-indol-2-yl)formamido]butanamide
(1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-yl)methanol
N-cyclopentyl-2-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,3-thiazole-4-carboxamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-[3-(1,2-oxazinan-2-yl)propanoyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
1-({5-[(3-fluoro-2,4-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propanamide
(1R,2R)-N-cyclopropyl-2-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropane-1-carboxamide
2-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-5-methyl-1H-1,3-benzodiazole
5-(2-fluorophenyl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
4-(4-chlorophenyl)-1-(1-ethyl-3-methylpiperidine-3-carbonyl)piperidin-4-ol
8-{6-carboxy-5-methylthieno[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-phenylacetamide
2-(morpholin-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
4-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-1,2-dihydropyridin-2-one
3-(3,4-dimethoxyphenyl)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpropanamide
8-(2-aminopyridine-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aR,7aS)-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide