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N-[(3-hydroxypyrrolidin-3-yl)methyl]-4-propylpyrimidine-5-carboxamide
ethyl 1-[2-(2,4-dioxo-1,3-thiazolidin-3-yl)acetyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
1-methyl-4-[5-methyl-6-(2-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]piperazine
4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,3-thiazole-5-carboxamide
N-cyclopropyl-6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[(2-chlorophenyl)methyl]-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]morpholine
5-(4-ethylpiperazine-1-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)morpholine-2-carboxamide
{4-[(4-chlorophenyl)methyl]-1-(2-methoxy-5-methylbenzenesulfonyl)piperidin-4-yl}methanol
4-(3,3-dimethyl-4-phenylpyrrolidin-1-yl)-4-oxobutane-1-sulfonamide
methyl 4-{[(1S,4S)-5-(3-chlorophenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}benzoate
4-[3-(cyclopropylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-6-fluoro-1,2,3,4-tetrahydroquinolin-2-one
4-[(2-chlorophenyl)methyl]-7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
{2,4,6-trimethyl-3-[({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)methyl]phenyl}methanol
2-[2-(4-chlorophenyl)morpholin-4-yl]-N-cyclopropylpyridine-4-carboxamide
{3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
3-cyclohexyl-2-oxo-1-(oxolan-2-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
methyl (2S)-2-{[5-(cycloheptylcarbamoyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridin-3-yl]formamido}-3-methylbutanoate
4,5-dimethyl-6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-2-(trifluoromethyl)pyrimidine
N-cyclohexyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(prop-2-yn-1-yl)propanamide
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-1-methyl-1H-imidazole-2-carboxamide
5-[1-(2-phenylethyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-benzyl[(1-oxo-2,3,4,9-tetrahydro-1H-carbazol-7-yl)amino]sulfonamide
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-[2-(pyridin-3-yloxy)ethyl]piperidin-4-amine
3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-(2,4,4-trimethylpentan-2-yl)piperidine-1-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-(5-phenyl-1,2,4-oxadiazol-3-yl)-3,6-diazabicyclo[3.2.2]nonane
5-methyl-N-(2-phenylpropyl)-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-{1-[6-(1H-indol-3-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
3-(1H-pyrazol-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-(cyclopentylamino)-4-methylpentane-1,4-diol
3-[(2-chlorophenyl)methyl]-N-methyl-N-(pyridin-2-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-{1-[3-(diethylamino)propanoyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-(1,3-thiazole-4-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N3-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
N-cyclobutyl-4-[methyl(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
1-(4-phenylpiperazin-1-yl)-3-{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}propan-1-one
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-3,5-dimethyl-1,2-oxazole-4-sulfonamide
6-cyclopentyl-1-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethan-1-one
2-{5-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
9-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(2S,4S)-1-benzyl-N-ethyl-4-{[(4-ethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
methyl 6-[2-(2-chloro-6-fluorophenyl)acetyl]-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1H-indole
2-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-2,3-dihydro-1,2-benzothiazol-3-one
ethyl 2-(4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-3-yl)acetate