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3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
(4aR,7aS)-1-propyl-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2R,3R)-1'-(2H-1,3-benzodioxol-5-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-(3-hydroxypiperidin-1-yl)ethan-1-one
5-(3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
4-[(4-ethoxyphenyl)methyl]-3-{2-oxo-2-[4-(pyridin-4-yl)piperazin-1-yl]ethyl}piperazin-2-one
5-methoxy-2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenol
5-chloro-2-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
N-[(1-cyclopentylpiperidin-4-yl)methyl]-6-oxo-N-(pyridin-3-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
3-benzyl-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxylic acid
1-(4,7-dimethylquinazolin-2-yl)-N-[1-(thiophen-2-yl)ethyl]piperidine-4-carboxamide
6-chloro-2-{1-[(5-methylpyrazin-2-yl)methyl]-1H-imidazol-2-yl}quinoline
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
2-methyl-5-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
3-[({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate
N-[3-(1H-imidazol-1-yl)butyl]-2,7,8-trimethylquinoline-4-carboxamide
ethyl 2-(2-{[1-(2-cyclohexylethyl)-1H-1,2,3-triazol-4-yl]formamido}ethyl)-1,3-thiazole-4-carboxylate
[2-(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenyl]methanol
N-(1H-imidazol-2-ylmethyl)-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(3-methyl-1-benzofuran-2-yl)methyl]acetamide
({5-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(3-methoxyphenyl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
methyl 1-ethyl-5-({[4-(methylsulfanyl)phenyl]methyl}amino)-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
propan-2-yl 2-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
(1R,3S)-3-(2-aminoethoxy)-7-(2-cyclopropylpyrimidine-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-cyclohexyl-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-methyl-4-phenyl-3-[1-(piperidine-1-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(2-ethoxyphenyl)methyl]-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-6-methylpyridine-2-carboxamide
2-(2-methoxyethyl)-9-(pyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
8-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(4-methylphenyl)methyl]-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazin-2-one
2-(3,4-dichlorophenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]morpholine
N-methyl-3-(propan-2-yl)-N-(quinolin-6-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
5-[(2S)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]pyrrolidin-2-yl]-3-methyl-1,2,4-oxadiazole
7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-ethylpiperidin-3-yl]methanol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
5-ethyl-3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-1,2,4-oxadiazole
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
5-(1H-1,3-benzodiazole-5-carbonyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N4-benzyl-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
8-({2-[(4-chlorophenyl)methoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)butan-1-one
(1H-imidazol-2-ylmethyl)({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
{4-[(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
(1S,5R)-N-(5-chloro-2-methoxyphenyl)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide