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2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]acetamide
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
6-(2,5-dimethylfuran-3-yl)-N-(2-hydroxybutyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[3-(1H-indol-1-yl)propyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-[(3R,4S)-1-(cyclopropylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-(1H-pyrazol-4-yl)propanamide
2-[3-(2,5-difluorophenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
6-chloro-2-[4-(5-methyl-1,3-oxazole-4-carbonyl)-1,4-diazepan-1-yl]-1,3-benzothiazole
3-(piperidin-1-ylmethyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-ol
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
(3R,4S)-3,4-dimethyl-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-4-ol
1-(2-fluorophenyl)-4-[1-(pentan-3-yl)piperidin-3-yl]piperazine
4-cyclopentyl-6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
N-[1-(2-methoxyphenoxy)propan-2-yl]-2-(methylamino)pyrimidine-5-carboxamide
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-N-(3,4-dimethylphenyl)piperidin-3-amine
1-(1-methylcyclopropanecarbonyl)-3-(2-phenylethyl)piperidine
methyl 5-[(4-hydroxybutan-2-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(4,4,4-trifluorobutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[(3,4-difluorophenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
7-(cyclohexylmethyl)-2-(4-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decane
1-methyl-N-[2-(2-methylphenoxy)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]amine
5-ethyl-3-({2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
[1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
benzyl 3-(4-chloro-1-methyl-1H-pyrazole-3-amido)pyrrolidine-1-carboxylate
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyrrolidin-3-yl)piperazine
1-[(2-chlorophenyl)methyl]-7-methoxy-3-({[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N2-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
1,9-dimethyl-4-(3-methyl-1-benzothiophene-2-carbonyl)-1,4,9-triazaspiro[5.5]undecane
N-(furan-3-ylmethyl)-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(3-methylphenoxy)piperidine
3-(4-hydroxyphenyl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H-pyrazole-5-carboxamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methoxybenzoyl)piperidine
(3aR,6aR)-2-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methoxy-N-[2-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methyl-1,3-thiazole-5-carboxamide
4-[4-(morpholin-4-yl)phenyl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-N-methylpyrimidin-2-amine
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-({7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
9-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-methoxy-N-{[1-(quinoline-6-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
3-(2-amino-1,3-thiazol-4-yl)-1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]propan-1-one
(3S,4S)-4-(4-fluorophenyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-ol
5-butyl-4-(2-hydroxyacetyl)-1-(3-phenylphenyl)piperazin-2-one
(3aS,6aR)-5-{[3-(methylsulfanyl)phenyl]methyl}-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(3,5-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one