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1-[(3-fluorophenyl)methyl]-4-(3-methoxy-5-methylthiophene-2-carbonyl)piperazine
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-phenoxybutan-1-one
2-(4-benzyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
N-[(3-chloro-2-fluorophenyl)methyl]-2-(morpholin-2-yl)acetamide
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine
1-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propan-1-ol
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
1-(4-tert-butylbenzoyl)-4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1,4-diazepan-5-one
1-phenyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)methanesulfonamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-azaspiro[5.5]undecan-9-amine
N-(1,3-benzothiazol-2-ylmethyl)-2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
2-methoxy-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]quinoline-4-carboxamide
N-(1-benzylpyrrolidin-3-yl)-2-methyl-2-(thiophen-2-ylformamido)propanamide
4-(1H-imidazol-1-ylmethyl)-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-ol
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[5-(trifluoromethyl)pyridin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-({4-[3-(5-methylfuran-2-yl)butyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-({7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
3-(1H-indol-3-ylmethyl)-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-oxo-N-{3-[(pyridin-3-yl)amino]propyl}-1,2-dihydroquinoline-4-carboxamide
5-methyl-6-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)thieno[2,3-d]pyrimidin-4-amine
2-[4-(2,6-diaminopyrimidin-4-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-methyl-4-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1-propyl-1H-pyrazole
(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
2-[(4-methoxyphenyl)methyl]-N-[1-(pyrimidin-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(2S)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}azetidine-2-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyridin-2-amine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(3S,4R)-1-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
3-(methylsulfanyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
1-{5-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-2-methoxyphenoxy}-3-(piperidin-1-yl)propan-2-ol
N-[1-(thian-4-yl)piperidin-4-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
3-(1,2-oxazinan-2-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(2-hydroxyethyl)piperidin-3-yl]propanamide
2-[(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]propanamide
2-{2-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,5-dimethyl-1H-1,3-benzodiazole
(2S,4S)-4-amino-1-(dimethyl-1,3-thiazole-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
2-(3-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)acetamide
3-[2-fluoro-3-(trifluoromethyl)phenyl]-1-(oxan-4-ylmethyl)urea
9-methoxy-N-[(3-methoxyphenyl)methyl]-3-[3-(methylsulfanyl)propanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[(3-methylphenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[1-(4-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]furan-3-carboxamide
2-methoxy-N-[(2R,3R)-1'-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide