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2-(1-methylpyrrolidin-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
9-(oxolane-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-[(2-aminopyridin-3-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(2S)-2-({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)-4-methylpentanamide
N-cyclohexyl-2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-(prop-2-yn-1-yl)acetamide
(1S,5R)-6-[3-(1H-pyrazol-1-yl)benzoyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-benzyl-8-[(5-methylfuran-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(azepan-1-yl)-2-phenylethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(cyclopropylmethyl)-5-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-methyl-4-({2-[3-(3-methylpiperidin-1-yl)propoxy]phenyl}methyl)piperazine
1-(2-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-cyclopropyl-9-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(5-chloropyridin-2-yl)-4-(1,3-thiazole-4-carbonyl)piperazine
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-3-(2-methyl-1H-indol-1-yl)propanamide
4-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine-2-carbonyl]morpholine
8-{[2-(methylsulfanyl)phenyl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-methyl-3-(pyridin-2-yl)-N-(thiolan-3-yl)-1H-pyrazol-5-amine
2-{4-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyrimidine
3-[(3R,4S)-1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
4-[(3-{5-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenyl)methyl]morpholine
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-methylfuran-2-carboxamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyridin-2-yl)ethan-1-one
2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-1-[4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
dimethyl({[(1R,5S,6S)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
8-methyl-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-methyl-3-(morpholin-4-yl)propan-1-one
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrrolidin-3-yl)benzamide
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-methoxy-5-methylphenyl)urea
1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[3-(dimethylamino)propyl]-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
7-[2-(methylsulfanyl)pyridine-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(3-{[1-(4-methoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
4-cyclopentyl-N-[1-(5-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
N-(4-{[(3S,4S)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-1-yl]methyl}phenyl)acetamide
1,5-dimethyl-4-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
[(4-methanesulfonylphenyl)methyl](methyl)[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
6-{octahydropyrrolo[1,2-a]piperazin-2-yl}-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
N,N-dimethyl-4-[(1E)-3-[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]prop-1-en-1-yl]aniline
methyl 5-[(1R,3S,4S)-3-hydroxy-4,7,7-trimethylbicyclo[2.2.1]heptane-1-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amine
6-ethyl-1-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(2-methoxyethyl)-4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepane-1-carbaldehyde
(1S,6R)-9-[3-(1H-pyrazol-1-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
1-(2H-1,3-benzodioxol-5-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
1-ethyl-3-[4-(morpholin-4-ylmethyl)phenyl]-1-[(2E)-3-phenylprop-2-en-1-yl]urea