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2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
8-chloro-3-(2-ethoxyphenyl)-[1,2,4]triazolo[4,3-a]pyridine
3-(3-chloro-1,2-oxazol-5-yl)-N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]propanamide
7-(2-methoxyethyl)-2-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[3-({7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenyl]ethan-1-one
2-(cyclopropylamino)-N-[phenyl(pyridin-4-yl)methyl]acetamide
N-methyl-N-(oxolan-3-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[3-(4-fluorophenoxy)propyl]-4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridine
methyl 5-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-5-oxopentanoate
ethyl 4-{[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}piperidine-1-carboxylate
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(3-methoxypropyl)piperidine
5-chloro-4,6-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
{4-[(5-methyl-4-phenyl-1H-imidazol-1-yl)methyl]phenyl}methanol
4-methyl-3-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzamide
(2E)-1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
[(3R,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
(2S)-3-methyl-2-[(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]butanamide
methyl 3-{[(2E)-3-(3-fluorophenyl)prop-2-enamido]methyl}-5-(thiophene-2-sulfonamido)benzoate
1-[2-(difluoromethoxy)benzoyl]-3-(3-methylphenoxy)azetidine
2-{9-[(5-fluoro-2-methoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
2-({7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)benzoic acid
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(1-methylpiperidin-4-yl)acetamide
2-chloro-N-(1,4-dioxan-2-ylmethyl)-5-(trifluoromethyl)benzamide
[(3R,4R)-1-(5-methoxyfuran-2-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
1-methyl-8-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(2,3-difluoro-4-methylphenyl)methyl]-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-(propan-2-yl)-5-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidine
3-[5-(5-methylpyrazine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(propan-2-yl)propanamide
1-[(2-fluorophenyl)methyl]-4-[2-(thiophen-3-yl)acetyl]piperazin-2-one
3-methyl-6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]pyridazine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(thiophene-3-sulfonyl)piperidine-3-carboxylate
(3R,4R)-1-[(2,3-difluoro-4-methylphenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-(dimethylamino)-N-[(5-ethylpyridin-2-yl)methyl]-2-(2-fluorophenyl)-N-methylacetamide
N-(1H-imidazol-2-ylmethyl)-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-6,8-dimethyl-2-(1H-pyrazol-4-yl)quinoline
6-[(1-benzylpiperidin-4-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(2,3-dihydro-1H-inden-1-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
(1R,7S)-3-(3-methylbutyl)-6-(5-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazole
3-{[7-(5-ethylthiophene-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridine-3-carboxamide
(2S)-2,6-diamino-N-(3-phenylprop-2-yn-1-yl)-N-propylhexanamide
1-(2-fluoro-5-methylphenyl)-3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}urea
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]urea
2-methyl-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide